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The discovery of equipotent PPARalpha/gamma dual activators.

Authors :
Martres P
Faucher N
Laroze A
Pineau O
Fouchet MH
Potvain F
Grillot D
Beneton V
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2008 Dec 01; Vol. 18 (23), pp. 6251-4. Date of Electronic Publication: 2008 Oct 01.
Publication Year :
2008

Abstract

We report the design and synthesis of equipotent PPARalpha/gamma dual agonists starting from selective PPAR alpha agonist 1. In vivo data for 7 in the Zucker fa/fa rat are presented.

Details

Language :
English
ISSN :
1464-3405
Volume :
18
Issue :
23
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
18947994
Full Text :
https://doi.org/10.1016/j.bmcl.2008.09.094