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Efficient C2 functionalisation of 2H-2-imidazolines.

Authors :
Bon RS
Sprenkels NE
Koningstein MM
Schmitz RF
de Kanter FJ
Dömling A
Groen MB
Orru RV
Source :
Organic & biomolecular chemistry [Org Biomol Chem] 2008 Jan 07; Vol. 6 (1), pp. 130-7. Date of Electronic Publication: 2007 Nov 08.
Publication Year :
2008

Abstract

Alkylation and oxidation of 2H-2-imidazolines, followed by regioselective deprotection, thionation and microwave-assisted Liebeskind-Srogl reaction, efficiently led to 2-aryl-2-imidazolines as new analogues of p53-hdm2 interaction inhibitors (Nutlins).

Details

Language :
English
ISSN :
1477-0520
Volume :
6
Issue :
1
Database :
MEDLINE
Journal :
Organic & biomolecular chemistry
Publication Type :
Academic Journal
Accession number :
18075657
Full Text :
https://doi.org/10.1039/b713065a