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An enantioselective Brønsted acid catalyzed enamine Mannich reaction.

Authors :
Tillman AL
Dixon DJ
Source :
Organic & biomolecular chemistry [Org Biomol Chem] 2007 Feb 21; Vol. 5 (4), pp. 606-9. Date of Electronic Publication: 2006 Dec 22.
Publication Year :
2007

Abstract

An enantioselective Brønsted acid catalyzed Mannich reaction between acetophenone derived enamines and N-Boc imines has been developed. Simple diol (S)-H(8)-BINOL has been identified as the optimal catalyst, to afford versatile beta-amino aryl ketones in good yield and enantiomeric excess.

Details

Language :
English
ISSN :
1477-0520
Volume :
5
Issue :
4
Database :
MEDLINE
Journal :
Organic & biomolecular chemistry
Publication Type :
Academic Journal
Accession number :
17285167
Full Text :
https://doi.org/10.1039/b616143j