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Unique tandem Heck-lactamization naphthyridinone ring formation between acrylanilides and halogenated pyridines.

Authors :
Cvetovich RJ
Reamer RA
DiMichele L
Chung JY
Chilenski JR
Source :
The Journal of organic chemistry [J Org Chem] 2006 Oct 27; Vol. 71 (22), pp. 8610-3.
Publication Year :
2006

Abstract

The Heck coupling of acrylanilides with 4-bromo-2-chloro-3-iodo-pyridine using palladium acetate can produce bis-Heck products or undergo an unusual tandem Heck-lactamization ring formation to generate 5-chloro-1-aryl-1,6-naphthyridin-2(1H)-ones.

Details

Language :
English
ISSN :
0022-3263
Volume :
71
Issue :
22
Database :
MEDLINE
Journal :
The Journal of organic chemistry
Publication Type :
Academic Journal
Accession number :
17064040
Full Text :
https://doi.org/10.1021/jo0613479