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Synthesis of 2-alkoxy-8-hydroxyadenylpeptides: towards synthetic epitope-based vaccines.

Authors :
Weterings JJ
Khan S
van der Heden GJ
Drijfhout JW
Melief CJ
Overkleeft HS
van der Burg SH
Ossendorp F
van der Marel GA
Filippov DV
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2006 Jun 15; Vol. 16 (12), pp. 3258-61. Date of Electronic Publication: 2006 Apr 11.
Publication Year :
2006

Abstract

The preparation of three different 2-alkoxy-8-hydroxyadenylpeptide conjugates has been accomplished by solid-phase synthesis combined with 'on-resin' Cu(I) catalyzed Huisgen cycloaddition. The immunogenicity of the compounds has been evaluated in IL-12 production and antigen presentation assays.

Details

Language :
English
ISSN :
0960-894X
Volume :
16
Issue :
12
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
16581248
Full Text :
https://doi.org/10.1016/j.bmcl.2006.03.034