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A switch in enantiomer preference between mitochondrial F1F0-ATPase chemotypes.

Authors :
Bisaha SN
Malley MF
Pudzianowski A
Monshizadegan H
Wang P
Madsen CS
Gougoutas JZ
Stein PD
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2005 Jun 02; Vol. 15 (11), pp. 2749-51.
Publication Year :
2005

Abstract

The preferred absolute configuration of two series of F(1)F(0)-ATP synthase inhibitors was determined. Although the configuration of the active enantiomer in each series is different, each series presents the same 'triaryl' pharmacophore to the enzyme binding site.

Details

Language :
English
ISSN :
0960-894X
Volume :
15
Issue :
11
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
15878269
Full Text :
https://doi.org/10.1016/j.bmcl.2005.03.115