Back to Search Start Over

Double diastereoselective [3,3]-sigmatropic aza-Claisen rearrangements.

Authors :
Davies SG
Garner AC
Nicholson RL
Osborne J
Savory ED
Smith AD
Source :
Chemical communications (Cambridge, England) [Chem Commun (Camb)] 2003 Sep 07 (17), pp. 2134-5.
Publication Year :
2003

Abstract

Asymmetric [3,3]-sigmatropic aza-Claisen rearrangement of the (Z)-N-allyl-N,O-silylketene aminal of (3S,4E,alphaR)-1-benzyloxy-3-(N-propionyl-N-alpha-methylbenzylamino)hex-4-ene furnishes (2S,3R,4E,alphaR)-N-alpha-methylbenzyl-2,3-dimethyl-7-benzyloxyhept-4-enamide in > 92% d.e.; rearrangement of the diastereomeric (3R,4E,alphaR)-(Z)-N,O-silylketene aminal proceeds with low diastereoselectivity.

Details

Language :
English
ISSN :
1359-7345
Issue :
17
Database :
MEDLINE
Journal :
Chemical communications (Cambridge, England)
Publication Type :
Academic Journal
Accession number :
13678167
Full Text :
https://doi.org/10.1039/b306323m