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Synthesis and biological evaluation of a new trioxaquine containing a trioxane moiety obtained by halogenocyclisation of a hemiperoxyacetal

Authors :
Dechy-Cabaret, Odile
Benoit-Vical, Françoise
Robert, Anne
Magnaval, Jean-François
Séguéla, Jean-Paul
Meunier, Bernard
Source :
Comptes Rendus Chimie. Jan2003, Vol. 6 Issue 1, p153. 8p.
Publication Year :
2003

Abstract

The preparation and the biological evaluation of a new antimalarial modular drug, named trioxaquine are reported. The trioxane moiety of this trioxaquine is prepared through the halogenocyclisation of a hemiperoxyacetal derived from the allylic hydroperoxide of 2,3-dimethyl-2-butene. [Copyright &y& Elsevier]

Details

Language :
English
ISSN :
16310748
Volume :
6
Issue :
1
Database :
Academic Search Index
Journal :
Comptes Rendus Chimie
Publication Type :
Academic Journal
Accession number :
9791240
Full Text :
https://doi.org/10.1016/S1631-0748(03)00007-9