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Total Synthesis and Antidepressant Activities of Laetispicine and Its Derivatives.

Authors :
Shuyi Yao
Hui Xie
Li Zhang
Tao Meng
Yongliang Zhang
Xin Wang
Lin Chen
Shengli Pan
Jingkang Shen
Source :
Molecules. Feb2012, Vol. 17 Issue 2, p1425-1436. 47p. 7 Diagrams, 1 Graph.
Publication Year :
2012

Abstract

The first total synthesis of laetispicine (1a), an amide alkaloid isolated from the stems of Piper laetispicum C.DC (Piperaceae), and the synthesis of some of its derivatives were described. Based on the evaluation of antidepressant activities in the forced swimming test, compounds 1h and 1i were identified as potent and safe antidepressant lead compounds. [ABSTRACT FROM AUTHOR]

Details

Language :
English
ISSN :
14203049
Volume :
17
Issue :
2
Database :
Academic Search Index
Journal :
Molecules
Publication Type :
Academic Journal
Accession number :
72015109
Full Text :
https://doi.org/10.3390/molecules17021425