Back to Search Start Over

Amplification of Screening Sensitivity through Selective Destruction: Theory and Screening of a Library of Carbonic Anhydrase Inhibitors.

Authors :
Cheeseman, Jeremy D.
Corbett, Andrew D.
Ronghua Shu
Croteau, Jonathan
Gleason, James L.
Kazlauskas, Romas J.
Source :
Journal of the American Chemical Society. 5/22/2002, Vol. 124 Issue 20, p5692. 10p. 6 Diagrams, 1 Chart, 11 Graphs.
Publication Year :
2002

Abstract

Assesses the screening method for the identification of enzyme inhibitors. Advantages of dynamic combinatorial chemistry; Suppression of carbonic anhydrase activity by sulfonamide dipeptides; Degradation of the poor inhibitors by enzymes.

Details

Language :
English
ISSN :
00027863
Volume :
124
Issue :
20
Database :
Academic Search Index
Journal :
Journal of the American Chemical Society
Publication Type :
Academic Journal
Accession number :
7060041
Full Text :
https://doi.org/10.1021/ja017099+