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2-Arylbenzoxazoles as novel cholesteryl ester transfer protein inhibitors: Optimization via array synthesis

Authors :
Harikrishnan, Lalgudi S.
Kamau, Muthoni G.
Herpin, Timothy F.
Morton, George C.
Liu, Yalei
Cooper, Christopher B.
Salvati, Mark E.
Qiao, Jennifer X.
Wang, Tammy C.
Adam, Leonard P.
Taylor, David S.
Chen, Alice Ye A.
Yin, Xiaohong
Seethala, Ramakrishna
Peterson, Tara L.
Nirschl, David S.
Miller, Arthur V.
Weigelt, Carolyn A.
Appiah, Kingsley K.
O’Connell, Jonathan C.
Source :
Bioorganic & Medicinal Chemistry Letters. Apr2008, Vol. 18 Issue 8, p2640-2644. 5p.
Publication Year :
2008

Abstract

Abstract: 2-Arylbenzoxazole 5 was identified as a hit from a fluorescence-based high-throughput screen for CETP inhibitors. The synthesis and SAR investigation employing array synthesis of the A- and B-rings are described. [Copyright &y& Elsevier]

Details

Language :
English
ISSN :
0960894X
Volume :
18
Issue :
8
Database :
Academic Search Index
Journal :
Bioorganic & Medicinal Chemistry Letters
Publication Type :
Academic Journal
Accession number :
31677410
Full Text :
https://doi.org/10.1016/j.bmcl.2008.03.030