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Substituted coumarins as potent 5-lipoxygenase inhibitors

Authors :
Grimm, Erich L.
Brideau, Christine
Chauret, Nathalie
Chan, Chi-Chung
Delorme, Daniel
Ducharme, Yves
Ethier, Diane
Falgueyret, Jean-Pierre
Friesen, Richard W.
Guay, Jocelyne
Hamel, Pierre
Riendeau, Denis
Soucy-Breau, Chantal
Tagari, Philip
Girard, Yves
Source :
Bioorganic & Medicinal Chemistry Letters. May2006, Vol. 16 Issue 9, p2528-2531. 4p.
Publication Year :
2006

Abstract

Abstract: Leukotriene biosynthesis inhibitors have potential as therapeutic agents for asthma and inflammatory diseases. A novel series of substituted coumarin derivatives has been synthesized and the structure–activity relationship was evaluated with respect to their ability to inhibit the formation of leukotrienes via the human 5-lipoxygenase enzyme. [Copyright &y& Elsevier]

Details

Language :
English
ISSN :
0960894X
Volume :
16
Issue :
9
Database :
Academic Search Index
Journal :
Bioorganic & Medicinal Chemistry Letters
Publication Type :
Academic Journal
Accession number :
20184167
Full Text :
https://doi.org/10.1016/j.bmcl.2006.01.085