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Palladium‐Catalyzed Carbonylative Difunctionalization of C=N Bond of Azaarenes or Imines to Quinazolinones.
- Source :
-
Chemistry - An Asian Journal . 6/2/2020, Vol. 15 Issue 11, p1678-1682. 5p. - Publication Year :
- 2020
-
Abstract
- Supporting information for this article is given via a link at the end of the document. By intercepting the acylpalladium species with C=N bond of azaarenes or imines other than free amines or alcohols, the difunctionalization of C=N bond was established via palladium‐catalyzed carbonylation/nucleophilic addition sequence. This method is compatible with a diverse range of azaarenes and imines and allows for the efficient synthesis of a wide range of quinazolinones and derivatives. The synthetic utility has been demonstrated by one‐step synthesis of evodiamine and its analogue with inexpensive starting materials. [ABSTRACT FROM AUTHOR]
- Subjects :
- *QUINAZOLINONES
*AZAARENES
*IMINES
*CARBONYLATION
*AMINES
*ALDIMINES
Subjects
Details
- Language :
- English
- ISSN :
- 18614728
- Volume :
- 15
- Issue :
- 11
- Database :
- Academic Search Index
- Journal :
- Chemistry - An Asian Journal
- Publication Type :
- Academic Journal
- Accession number :
- 143547818
- Full Text :
- https://doi.org/10.1002/asia.202000359