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Estrogen receptor ligands. Part 1: The discovery of flavanoids with subtype selectivity

Authors :
Chen, Helen Y.
Dykstra, Kevin D.
Birzin, Elizabeth T.
Frisch, Katalin
Chan, Wanda
Yang, Yi T.
Mosley, Ralph T.
DiNinno, Frank
Rohrer, Susan P.
Schaeffer, James M.
Hammond, Milton L.
Source :
Bioorganic & Medicinal Chemistry Letters. Mar2004, Vol. 14 Issue 6, p1417. 5p.
Publication Year :
2004

Abstract

A class of flavanoids exhibiting a high degree of selectivity for ERα over ERβ has been discovered. The most active analogue 6 was found to be 66-fold ERα-selective and demonstrated uterine estradiol antagonism. [Copyright &y& Elsevier]

Details

Language :
English
ISSN :
0960894X
Volume :
14
Issue :
6
Database :
Academic Search Index
Journal :
Bioorganic & Medicinal Chemistry Letters
Publication Type :
Academic Journal
Accession number :
12433655
Full Text :
https://doi.org/10.1016/j.bmcl.2004.01.031