198 results on '"Yusuf Özkay"'
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2. Synthesis, DFT Calculations, In Silico Studies, and Antimicrobial Evaluation of Benzimidazole-Thiadiazole Derivatives
3. New Benzimidazole-Triazole Derivatives as Topoisomerase I Inhibitors: Design, Synthesis, Anticancer Screening, and Molecular Modeling Studies
4. Design, Synthesis, and Biological Effect Studies of Novel Benzofuran–Thiazolylhydrazone Derivatives as Monoamine Oxidase Inhibitors
5. Synthesis and Anticancer Activities of Pyrazole–Thiadiazole-Based EGFR Inhibitors
6. Design, Synthesis, and Biological Evaluation Studies of Novel Naphthalene-Chalcone Hybrids As Antimicrobial, Anticandidal, Anticancer, and VEGFR‑2 Inhibitors
7. Investigation of Novel Quinoline–Thiazole Derivatives as Antimicrobial Agents: In Vitro and In Silico Approaches
8. Synthesis, Molecular Docking, Dynamics, Quantum-Chemical Computation, and Antimicrobial Activity Studies of Some New Benzimidazole–Thiadiazole Hybrids
9. Synthesis, in vitro enzyme activity and molecular docking studies of new benzylamine-sulfonamide derivatives as selective MAO-B inhibitors
10. Synthesis, anticancer evaluation and molecular docking studies of new benzimidazole- 1,3,4-oxadiazole derivatives as human topoisomerase types I poison
11. Design, Synthesis, and Evaluation of Novel 2H-Benzo[b][1,4]thiazin-3(4H)-one Derivatives as New Acetylcholinesterase Inhibitors
12. Novel Thiosemicarbazone Derivatives: In Vitro and In Silico Evaluation as Potential MAO-B Inhibitors
13. Yeni piperazin bileşiklerinin sentezi ve antikolinesteraz etkilerinin araştırılması
14. 9th International Congress on Psychopharmacology & 5th International Symposium on Child and Adolescent Psychopharmacology
15. Design, synthesis, and evaluation of novel 2-phenylpropionic acid derivatives as dual COX inhibitory-antibacterial agents
16. Novel 1-(2-pyrimidin-2-yl)piperazine derivatives as selective monoamine oxidase (MAO)-A inhibitors
17. Design, Synthesis, and Structure–Activity Relationships of Thiazole Analogs as Anticholinesterase Agents for Alzheimer’s Disease
18. Design, Synthesis, In Vitro and In Silico Studies of New Thiazolylhydrazine-Piperazine Derivatives as Selective MAO-A Inhibitors
19. Design, Synthesis, and Biological Activity Evaluation of New Donepezil-Like Compounds Bearing Thiazole Ring for the Treatment of Alzheimer’s Disease
20. Synthesis, Docking Studies and Biological Activity of New Benzimidazole- Triazolothiadiazine Derivatives as Aromatase Inhibitor
21. Synthesis and Evaluation of N-[1-(((3,4-Diphenylthiazol-2(3H)-ylidene)amino)methyl)cyclopentyl]acetamide Derivatives for the Treatment of Diseases Belonging to MAOs
22. Synthesis, Molecular Docking Studies, and Antifungal Activity Evaluation of New Benzimidazole-Triazoles as Potential Lanosterol 14α-Demethylase Inhibitors
23. Synthesis and AChE Inhibitory Activity of Novel Thiazolylhydrazone Derivatives
24. Synthesis and Antifungal Potential of Some Novel Benzimidazole-1,3,4-Oxadiazole Compounds
25. Synthesis and Evaluation of New 1,3,4-Thiadiazole Derivatives as Potent Antifungal Agents
26. Synthesis and Biological Evaluation of Novel Piperazine Containing Hydrazone Derivatives
27. Synthesis and Biological Evaluation of New Cholinesterase Inhibitors for Alzheimer’s Disease
28. Synthesis of New Benzothiazole Acylhydrazones as Anticancer Agents
29. Design and Synthesis of New Benzothiazole Compounds as Selective hMAO-B Inhibitors
30. Synthesis and Biological Evaluation of New Thiosemicarbazone Derivative Schiff Bases as Monoamine Oxidase Inhibitory Agents
31. Synthesis and Anticandidal Activity Evaluation of New Benzimidazole-Thiazole Derivatives
32. Synthesis of Oxadiazole-Thiadiazole Hybrids and Their Anticandidal Activity
33. Synthesis of Some New Thiazole Derivatives and Their Biological Activity Evaluation
34. Synthesis of 2-(5-(2-((5-(Cyclohexylamino)-1,3,4-Thiadiazol-2-yl)thio)ethyl)-1,3,4-Oxadiazol-2-yl) Derivatives and Their Antimicrobial Activity
35. Synthesis and Antimicrobial Activity Evaluation of New Benzimidazole—Thiazole Derivatives
36. Synthesis and Anticandidal Activity of New Imidazole Derivatives
37. Synthesis and Antimicrobial Activity of Newly Synthesized 2-((5-(4-(5(6)fluoro-1H-benzo[d]imidazol-2-yl)phenyl)-1,3,4-oxadiazol-2-yl)thio)-Derivatives
38. Novel Imidazole Derivatives as Antifungal Agents: Synthesis, Biological Evaluation, ADME Prediction and Molecular Docking Studies
39. Synthesis, Anticandidal Activity and Molecular Docking Study of Some New Imidazole Derivatives
40. Design, Synthesis Molecular Docking Study and Antifungal Activity Evaluation of New Benzimidazole-Triazole Derivatives
41. Pharmacological and Toxicological Screening of Novel Benzimidazole-Morpholine Derivatives as Dual-Acting Inhibitors
42. Synthesis of New Hydrazone Derivatives for MAO Enzymes Inhibitory Activity
43. New Benzimidazole-1,2,4-Triazole Hybrid Compounds: Synthesis, Anticandidal Activity and Cytotoxicity Evaluation
44. Synthesis and Biological Evaluation of Some Novel Dithiocarbamate Derivatives
45. Synthesis, biological activity evaluation and molecular docking studies of novel thiazole derivatives
46. Thiazole inhibitors of α-glucosidase: Positional isomerism modulates selectivity, enzyme binding and potency of inhibition.
47. Design, Synthesis, and In Vitro and In Silico Approaches of Novel Indanone Derivatives as Multifunctional Anti-Alzheimer Agents
48. Synthesis of new compounds bearing methyl sulfonyl pharmacophore as selective <scp>COX</scp> ‐2 inhibitor
49. Synthesis of new derivatives containing pyridine, investigation of MAO inhibitory activities and molecular docking studies
50. Synthesis of Some 2-Substituted-5-(Benzothiazol-2-yl)-1H-Benzimidazole Derivatives and Investigation of Their Antiproliferative Effects
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