225 results on '"Vyas, Dolatrai M."'
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2. Pyrrolotriazine-5-carboxylate ester inhibitors of EGFR and HER2 protein tyrosine kinases and a novel one-pot synthesis of C-4 subsitituted pyrrole-2,3-dicarboxylate diesters (1)
3. Some Recent Developments in the Synthesis and Structure-Activity Relationship of Novel Taxanes
4. Synthesis and biological evaluation of C-13 amide-linked paclitaxel (Taxol) analogs
5. Recent Developments in Cancer Cytotoxics
6. The discovery of BMS-275183: an orally efficacious novel taxane
7. 6 Paclitaxel: A Unique Tubulin Interacting Anticancer Agent
8. Stereospecific synthesis of 7-deoxy-6-hydroxy paclitaxel
9. Proline isosteres in a series of 2,4-disubstituted pyrrolo[1,2- f][1,2,4]triazine inhibitors of IGF-1R kinase and IR kinase
10. ChemInform Abstract: Synthesis and Antitumor Activity of Novel Paclitaxel-Chlorambucil Hybrids.
11. ChemInform Abstract: Synthesis of 7β-Sulfur Analogues of Paclitaxel Utilizing a Novel Epimerization of the 7α-Thiol Group.
12. ChemInform Abstract: Oxime Derivatives of Sordaricin as Potent Antifungal Agents.
13. ChemInform Abstract: Nucleophilic Capture of the Imino-Quinone Methide Type Intermediates Generated from 2-Aminothiazol-5-yl Carbinols.
14. Nucleophilic Capture of the Imino-Quinone Methide Type Intermediates Generated from 2-Aminothiazol-5-yl Carbinols
15. Discovery and Preclinical Evaluation of [4-[[1-(3-fluorophenyl)methyl]-1H-indazol-5-ylamino]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl]carbamic Acid, (3S)-3-Morpholinylmethyl Ester (BMS-599626), a Selective and Orally Efficacious Inhibitor of Human Epidermal Growth Factor Receptor 1 and 2 Kinases
16. Discovery of a 2,4-Disubstituted Pyrrolo[1,2-f][1,2,4]triazine Inhibitor (BMS-754807) of Insulin-like Growth Factor Receptor (IGF-1R) Kinase in Clinical Development
17. 5-((4-Aminopiperidin-1-yl)methyl)pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases
18. Synthesis and structure–activity relationship of imidazo(1,2- a)thieno(3,2- e)pyrazines as IKK-β inhibitors
19. Novel C-5 aminomethyl pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases
20. New C-5 substituted pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases
21. Novel 1 H-(benzimidazol-2-yl)-1 H-pyridin-2-one inhibitors of insulin-like growth factor I (IGF-1R) kinase
22. Novel 1H-(benzimidazol-2-yl)-1H-pyridin-2-one inhibitors of insulin-like growth factor I (IGF-1R) kinase
23. New dual inhibitors of EGFR and HER2 protein tyrosine kinases
24. Chemotherapeutics, Anticancer
25. Novel 3‘,6‘-Anhydro and N12,N13-Bridged Glycosylated Fluoroindolo[2,3-a]carbazoles as Topoisomerase I Inhibitors. Fluorine as a Leaving Group from sp3Carbon
26. Discovery of a Fluoroindolo[2,3-a]carbazole Clinical Candidate with Broad Spectrum Antitumor Activity in Preclinical Tumor Models Superior to the Marketed Oncology Drug, CPT-11
27. Design and Synthesis of a Fluoroindolocarbazole Series as Selective Topoisomerase I Active Agents. Discovery of Water-Soluble 3,9-Difluoro-12,13-dihydro-13-[6-amino-β-d-glucopyranosyl]-5H,13H-benzo[b]thienyl[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6H)-dione (BMS-251873) with Curative Antitumor Activity against Prostate Carcinoma Xenograft Tumor Model.
28. Design and Synthesis of a Fluoroindolocarbazole Series as Selective Topoisomerase I Active Agents. Discovery of Water-Soluble 3,9-Difluoro-12,13-dihydro-13-[6-amino-β- d-glucopyranosyl]-5H,13H-benzo[b]- thienyl[2,3-a]pyrrolo[3,4-c]carbazole- 5,7(6H)-dione (BMS-251873) with Curative Antitumor Activity against Prostate Carcinoma Xenograft Tumor Model
29. Identification of a broad-Spectrum azasordarin with improved pharmacokinetic properties
30. Sordaricin antifungal agents
31. Core-modified sordaricin derivatives: Synthesis and antifungal activity
32. Sordarin Oxazepine Derivatives as Potent Antifungal Agents
33. Oxime derivatives of sordaricin as potent antifungal agents
34. 2-Aryl-2,2-difluoroacetamide FKBP12 Ligands: Synthesis and X-ray Structural Studies
35. Synthesis and Antitumor Activity of Novel C-7 Paclitaxel Ethers: Discovery of BMS-184476
36. Synthesis of 7β-Sulfur Analogues of Paclitaxel Utilizing a Novel Epimerization of the 7α-Thiol Group
37. Synthesis of metabolically blocked paclitaxel analogues
38. Synthesis and antitumor activity of novel paclitaxel–chlorambucil hybrids
39. Chemotherapeutics, Anticancer
40. Structure–activity relationships study at the 3′-N position of paclitaxel. part 2: synthesis and biological evaluation of 3′-N-thiourea- and 3′-N-thiocarbamate-bearing paclitaxel analogues
41. Stereospecific synthesis of the major human metabolite of paclitaxel
42. ChemInform Abstract: Stereospecific Synthesis of 7‐Deoxy‐6‐hydroxy Paclitaxel.
43. Synthesis of a paclitaxel isomer: C-2-acetoxy-C-4-benzoate paclitaxel
44. Crystallographic determination of the stereochemistry of C-6,7 epoxy paclitaxel
45. Synthesis of a hybrid analog of the esperamicin and dynemicin cores
46. Synthesis of an esperamicin core analog with an epoxide trigger
47. TAXOL®: Science and Applications Edited by Matthew Suffness (National Cancer Institute). CRC Press, Boca Raton, FL. 1995. xii + 426pp. 17.5 × 25 cm. $136.95. ISBN 0-8493-8382-X.
48. Novel C-4 paclitaxel (Taxol®) analogs: potent antitumor agents
49. The synthesis and biological activity of enediyne minor groove binding hybrids
50. Editorial
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