45 results on '"Traeger, Sarah C."'
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2. Synthesis of an adenine N-3 substituted CBI adduct by alkylation of adenine with a 1-iodomethylindoline seco-CBI precursor
3. Synthesis of Bicyclo[1.1.0]butanes from Iodo-Bicyclo[1.1.1]pentanes
4. Synthesis and biological evaluation of biaryl alkyl ethers as inhibitors of IDO1
5. The role of chromatographic and chiroptical spectroscopic techniques and methodologies in support of drug discovery for atropisomeric drug inhibitors of Bruton’s tyrosine kinase
6. Amination of Nitro-Substituted Heteroarenes by Nucleophilic Substitution of Hydrogen
7. Structural and Thermal Characterization of Halogenated Azidopyridines: Under-Reported Synthons for Medicinal Chemistry
8. Discovery of an Oxycyclohexyl Acid Lysophosphatidic Acid Receptor 1 (LPA1) Antagonist BMS-986278 for the Treatment of Pulmonary Fibrotic Diseases
9. Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Using Scaffold-Hopping and Structure-Guided Drug Design
10. Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 Inhibitors
11. Discovery of Imidazopyridines as Potent Inhibitors of Indoleamine 2,3-Dioxygenase 1 for Cancer Immunotherapy
12. Discovery and Preclinical Evaluation of BMS-986242, a Potent, Selective Inhibitor of Indoleamine-2,3-dioxygenase 1
13. Structural and Thermal Characterization of Halogenated Azidopyridines: Under-Reported Synthons for Medicinal Chemistry.
14. Identification of Reversible Small Molecule Inhibitors of Endothelial Lipase (EL) That Demonstrate HDL-C Increase In Vivo
15. Use of a Conformational-Switching Mechanism to Modulate Exposed Polarity: Discovery of CCR2 Antagonist BMS-741672
16. Evolution of a Scale-Up Synthesis to a Potent GluN2B Inhibitor and Its Prodrug
17. An efficient one-pot synthesis of substituted 2-aminobenzo-1-thiophene-3-carbonitriles
18. Discovery of 6-Fluoro-5-(R)-(3-(S)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4H)-yl)-2-methylphenyl)-2-(S)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxamide (BMS-986142): A Reversible Inhibitor of Bruton’s Tyrosine Kinase (BTK) Conformationally Constrained by Two Locked Atropisomers
19. ChemInform Abstract: An Efficient One‐Pot Synthesis of Substituted 2‐Aminobenzo‐1‐thiophene‐3‐carbonitriles.
20. Discovery of a Potent and Orally Bioavailable Dual Antagonist of CC Chemokine Receptors 2 and 5
21. Discovery of Potent Heterodimeric Antagonists of Inhibitor of Apoptosis Proteins (IAPs) with Sustained Antitumor Activity
22. From rigid cyclic templates to conformationally stabilized acyclic scaffolds. Part II: Acyclic replacements for the (3 S)-3-benzylpiperidine in a series of potent CCR3 antagonists
23. Confirmation That Cytochrome P450 2C8 (CYP2C8) Plays a Minor Role in (S)-(+)- and (R)-(-)-Ibuprofen Hydroxylation in Vitro
24. ChemInform Abstract: One-Pot Two Step Synthesis of 5-Cyano-dihydropyrimidinones Using Polyphosphate Ester.
25. One-pot two step synthesis of 5-cyano-dihydropyrimidinones using polyphosphate ester
26. From rigid cyclic templates to conformationally stabilized acyclic scaffolds. Part II: Acyclic replacements for the (3S)-3-benzylpiperidine in a series of potent CCR3 antagonists
27. Discovery of Potent HeterodimericAntagonists of Inhibitorof Apoptosis Proteins (IAPs) with Sustained Antitumor Activity.
28. Discovery and Development of 5-[(5S,9R)-9- (4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1- methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]non- 7-yl-methyl]-3-thiophenecarboxylic Acid (BMS-587101)A Small Molecule Antagonist of Leukocyte Function Associated Antigen-1
29. Synthesis and SAR of pyrrolotriazine-4-one based Eg5 inhibitors
30. Solid-Phase Synthesis of 5-Substituted Amino Pyrazoles
31. One‐Pot Synthesis and Conformational Features of N,N′‐Disubstituted Ketene Aminals.
32. One-Pot Synthesis and Conformational Features of N,N‘-Disubstituted Ketene Aminals
33. Design and Synthesis of 4-Substituted Benzamides as Potent, Selective, and Orally Bioavailable IKs Blockers
34. ChemInform Abstract: Efficient Molar-Scale Synthesis of 1-Methyl-5-acylimidazole Triflic Acid Salts.
35. Efficient Molar-Scale Synthesis of 1-Methyl-5-acylimidazole Triflic Acid Salts
36. Binding of ATP-Sensitive Potassium Channel (KATP) Openers to Cardiac Membranes: Correlation of Binding Affinities with Cardioprotective and Smooth Muscle Relaxing Potencies
37. Cardioselective Antiischemic ATP-Sensitive Potassium Channel (KATP) Openers. 5. Identification of 4-(N-Aryl)-Substituted Benzopyran Derivatives with High Selectivity
38. α-Phosphonosulfonic Acids: Potent and Selective Inhibitors of Squalene Synthase
39. Diastereoselective oxidation of sulfides to sulfoxides. Synthesis of novel C-6 sulfoxy tetrahydromevinic acids
40. 1,2,3,4-tetrahydro-8-hydroxymanzamines, alkaloids from two different haplosclerid sponges
41. Novel Bishomoscalarane Sesterterpenes from the Sponge Phyllospongia foliascens
42. One-Pot Synthesis and Conformational Features of N,N'-Disubstituted Ketene Aminals.
43. Discovery of an Oxycyclohexyl Acid Lysophosphatidic Acid Receptor 1 (LPA 1 ) Antagonist BMS-986278 for the Treatment of Pulmonary Fibrotic Diseases.
44. Discovery and development of 5-[(5S,9R)-9-(4-cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]non-7-yl-methyl]-3-thiophenecarboxylic acid (BMS-587101)--a small molecule antagonist of leukocyte function associated antigen-1.
45. One-pot synthesis and conformational features of n,n'-disubstituted ketene aminals.
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