203 results on '"Tomassi, Stefano"'
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2. Comprehensive structural investigation of a potent and selective CXCR4 antagonist via crosslink modification
3. Disulfide bond replacement with non-reducible side chain to tail macrolactamization for the development of potent and selective CXCR4 peptide antagonists endowed with flanking binding sites
4. Irreversible inhibition of TRF2TRFH recruiting functions by a covalent cyclic peptide induces telomeric replication stress in cancer cells
5. Ultrasound-assisted Peptide Nucleic Acids synthesis (US-PNAS)
6. Novel pyridine-containing histone deacetylase inhibitors strongly arrest proliferation, induce apoptosis and modulate miRNAs in cancer cells
7. Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models
8. The organometallic ferrocene exhibits amplified anti-tumor activity by targeted delivery via highly selective ligands to αvβ3, αvβ6, or α5β1 integrins
9. A combined approach of structure‐based virtual screening and NMR to interrupt the PD‐1/PD‐L1 axis: Biphenyl‐benzimidazole containing compounds as novel PD‐L1 inhibitors
10. Cationic nucleopeptides as novel non-covalent carriers for the delivery of peptide nucleic acid (PNA) and RNA oligomers
11. New insights in the structure-activity relationships of 2-phenylamino-substituted benzothiopyrano[4,3-d]pyrimidines as kinase inhibitors
12. A combined approach of structure‐based virtual screening and NMR to interrupt the PD‐1/PD‐L1 axis: Biphenyl‐benzimidazole containing compounds as novel PD‐L1 inhibitors.
13. Specific Inhibitors of Mitochondrial Deacylase Sirtuin 4 Endowed with Cellular Activity.
14. First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8
15. Irreversible inhibition of TRF2TRFHrecruiting functions: a strategy to induce telomeric replication stress in cancer cells
16. Tailoring the Structure of Cell Penetrating DNA and RNA Binding Nucleopeptides
17. Design and synthesis of Nrf2-derived hydrocarbon stapled peptides for the disruption of protein-DNA-interactions
18. CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists
19. A novel smaller β‐defensin‐derived peptide is active against multidrug‐resistant bacterial strains
20. Polycomb Repressive Complex 2 Modulation through the Development of EZH2–EED Interaction Inhibitors and EED Binders
21. Halting the Spread of Herpes Simplex Virus-1: The Discovery of an Effective Dual αvβ6/αvβ8 Integrin Ligand
22. Click-Chemistry (CuAAC) Trimerization of an αvβ₆ Integrin Targeting Ga-68-Peptide : Enhanced Contrast for in-Vivo PET Imaging of Human Lung Adenocarcinoma Xenografts
23. Novel Peptide-Based PET Probe for Non-invasive Imaging of C-X-C Chemokine Receptor Type 4 (CXCR4) in Tumors
24. Characterization of water-soluble esters of nitrobenzoxadiazole-based GSTP1-1 inhibitors for cancer treatment
25. Disulfide Bond Replacement with 1,4‐ and 1,5‐Disubstituted [1,2,3]‐Triazole on C‐X‐C Chemokine Receptor Type 4 (CXCR4) Peptide Ligands: Small Changes that Make Big Differences
26. Properly Substituted Cyclic Bis-(2-bromobenzylidene) Compounds Behaved as Dual p300/CARM1 Inhibitors and Induced Apoptosis in Cancer Cells
27. Click‐Chemistry (CuAAC) Trimerization of an αvβ6 Integrin Targeting Ga‐68‐Peptide: Enhanced Contrast for in‐Vivo PET Imaging of Human Lung Adenocarcinoma Xenografts
28. HOPPI-NMR: Hot-Peptide-Based Screening Assay for Inhibitors of Protein–Protein Interactions by NMR
29. From PARP1 to TNKS2 Inhibition: A Structure-Based Approach
30. From a Helix to a Small Cycle: Metadynamics-Inspired αvβ6 Integrin Selective Ligands
31. Boosting Fmoc Solid-Phase Peptide Synthesis by Ultrasonication
32. Investigation of the Stereochemical-Dependent DNA and RNA Binding of Arginine-Based Nucleopeptides
33. Discovery of Pyrido[3′,2′:5,6]thiopyrano[4,3-d]pyrimidine-Based Antiproliferative Multikinase Inhibitors
34. Click‐Chemistry (CuAAC) Trimerization of an αvβ6 Integrin Targeting Ga‐68‐Peptide: Enhanced Contrast for in‐Vivo PET Imaging of Human Lung Adenocarcinoma Xenografts.
35. Combined HAT/EZH2 modulation leads to cancer-selective cell death
36. Simultaneous Targeting of RGD-Integrins and Dual Murine Double Minute Proteins in Glioblastoma Multiforme
37. Von einer Helix zu einem kleinen Ring: Metadynamik-inspirierte, selektive Liganden für αvβ6-Integrin
38. From a Helix to a Small Cycle: Metadynamics-Inspired αvβ6 Integrin Selective Ligands
39. Antitumor efficacy of Kisspeptin in human malignant mesothelioma cells
40. Ligand-Based NMR Study of C-X-C Chemokine Receptor Type 4 (CXCR4)–Ligand Interactions on Living Cancer Cells
41. Phenotypic Identification of a Novel Autophagy Inhibitor Chemotype Targeting Lipid Kinase VPS34
42. Structure–Activity Relationships and Biological Characterization of a Novel, Potent, and Serum Stable C-X-C Chemokine Receptor Type 4 (CXCR4) Antagonist
43. Phenotypic Identification of a Novel Autophagy Inhibitor Chemotype Targeting Lipid Kinase VPS34
44. Indazole-Based Covalent Inhibitors To Target Drug-Resistant Epidermal Growth Factor Receptor
45. Structure–Activity Relationships and Biological Characterization of a Novel, Potent, and Serum Stable C-X-C Chemokine Receptor Type 4 (CXCR4) Antagonist
46. Design, synthesis and biological evaluation of small molecules as modulators of histone methyltransferases and demethylases
47. Switchable Protecting Strategy for Solid Phase Synthesis of DNA and RNA Interacting Nucleopeptides
48. Exploring the N-Terminal Region of C-X-C Motif Chemokine 12 (CXCL12): Identification of Plasma-Stable Cyclic Peptides As Novel, Potent C-X-C Chemokine Receptor Type 4 (CXCR4) Antagonists
49. Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach
50. Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach
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