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916 results on '"Structure–activity relationship (SAR)"'

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9. Design, Structure–Activity Relationships, and Computational Modeling Studies of a Series of α-Helix Biased, Ultra-Short Glucagon-like Peptide-1 Receptor Agonists.

10. Synthesis and biological evaluation of ortho-phenyl phenylhydroxamic acids containing phenothiazine with improved selectivity for class IIa histone deacetylases.

11. Structure–Tissue Exposure/Selectivity Relationship (STR) on Carbamates of Cannabidiol.

13. Boosting of retinol activity using novel lecithin: Retinol acyltransferase inhibitors.

14. Exploring Benzimidazole Chemistry: Synthesis, Biological activity, and Molecular Docking Studies for Alzheimer's Treatment.

15. A SAR and QSAR study on 3CLpro inhibitors of SARS-CoV-2 using machine learning methods.

16. Evaluation of the Therapeutic Potential of Sulfonyl Urea Derivatives as Soluble Epoxide Hydrolase (sEH) Inhibitors.

17. Recent pharmacological insights about imidazole hybrids: a comprehensive review.

18. Illuminating Potential of Diphenyltin(IV) Dithiocarbamate Compounds for Pharmacological Applications: Synthesis, Structural Elucidation, In-silico and Cytotoxicity Study on A549 Human Lung Cancer Cells.

21. A review on natural sweeteners, sweet taste modulators and bitter masking compounds: structure-activity strategies for the discovery of novel taste molecules.

22. SAR, Molecular Docking and Molecular Dynamic Simulation of Natural Inhibitors against SARS-CoV-2 Mpro Spike Protein.

23. Comparative structure activity and target exploration of 1,2-diphenylethynes in Haemonchus contortus and Caenorhabditis elegans

24. Synthesis and biological evaluation of C-4 substituted phenoxazine-bearing hydroxamic acids with potent class II histone deacetylase inhibitory activities.

25. Organometallic N‐acylhydrazones of 5‐nitrofuran and 5‐nitrothiophene based: Synthesis, electrochemical, antiparasitic evaluation, and computational study.

27. A critical review of benzimidazole: Sky-high objectives towards the lead molecule to predict the future in medicinal chemistry

28. Nonlinear SAR Modelling of Mosquito Repellents for Skin Application.

29. Current Advancements for New Drug Discovery Against Dengue Virus: A Review (2015 – 2020).

30. Investigation of the mechanism of action of mefloquine and derivatives against the parasite Echinococcus multilocularis

31. Structure-activity correlations for peptaibols obtained from clade Longibrachiatum of Trichoderma: A combined experimental and computational approach

32. Upregulation of p53 through induction of MDM2 degradation: improved potency through the introduction of an alkylketone sidechain on the anthraquinone core

33. Applications and Potential of In Silico Approaches for Psychedelic Chemistry.

34. Design, Synthesis, Computational and Biological Evaluation of Novel Structure Fragments Based on Lithocholic Acid (LCA).

35. CL-705G: a novel chemical Kir6.2-specific KATP channel opener.

36. Tunable Fluorescence via Self-Assembled Switching of AIE-Active Micelle-like Nanoaggregates.

37. Classification models and SAR analysis on HDAC1 inhibitors using machine learning methods.

38. CL-705G: a novel chemical Kir6.2-specific KATP channel opener

39. Design, Synthesis, and Evaluation of Niclosamide Analogs as Therapeutic Agents for Enzalutamide-Resistant Prostate Cancer.

40. Theonella : A Treasure Trove of Structurally Unique and Biologically Active Sterols.

41. A Lipidated Single-B-Chain Derivative of Relaxin Exhibits Improved In Vitro Serum Stability without Altering Activity.

42. Investigation of the mechanism of action of mefloquine and derivatives against the parasite Echinococcus multilocularis.

43. Design and synthesis of novel hydrazinyl thiazoles from biomass derived furfurals: Their molecular docking, anti-cancer, anti-oxidant, and anti-bacterial study.

44. Exploring the molecular insights of imidazole and benzimidazole scaffold for cancer therapy: Synthesis, in-vitro cytotoxicity and SAR studies.

45. Structure-activity relationship read-across and transcriptomics for branched carboxylic acids.

46. In Vitro and In Silico Biological Studies of 4-Phenyl-2-quinolone (4-PQ) Derivatives as Anticancer Agents.

47. Antifouling activity of terpenoids from the corals Sinularia flexibilis and Muricella sp. against the bryozoan Bugula neritina.

48. ANTICANCER POTENTIAL OF COMPOUNDS BEARING THIAZOLIDIN-4-ONE SCAFFOLD: COMPREHENSIVE REVIEW.

49. Resveratrol-like Compounds as SIRT1 Activators.

50. Upregulation of p53 through induction of MDM2 degradation: improved potency through the introduction of an alkylketone sidechain on the anthraquinone core.

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