1,081 results on '"Spring, David R."'
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2. Publisher Correction: Novel immunotherapeutics against LGR5 to target multiple cancer types
3. Selective Aurora A‑TPX2 Interaction Inhibitors Have In Vivo Efficacy as Targeted Antimitotic Agents.
4. Towards the Targeted Protein Degradation of PRMT1
5. CK2 Inhibitors Targeting Inside and Outside the Catalytic Box
6. Selective Aurora A-TPX2 Interaction Inhibitors Have In VivoEfficacy as Targeted Antimitotic Agents
7. Tuneable thiol exchange linkers for traceless drug release applications in prodrugs and ADCs.
8. Unlocking Amides: A General Method for the Self‐Immolative Release of Amide‐Containing Molecules
9. Site-selective peptide functionalisation mediated via vinyl-triazine linchpins
10. Red-light modulated ortho-chloro azobenzene photoswitch for peptide stapling via aromatic substitution
11. Microscopy and chemical analyses reveal flavone-based woolly fibres extrude from micron-sized holes in glandular trichomes of Dionysia tapetodes
12. Energetics of lipid transport by the ABC transporter MsbA is lipid dependent
13. Photoredox C(2)-Arylation of Indole- and Tryptophan-Containing Biomolecules.
14. Synthesis of structurally diverse biflavonoids
15. Novel non-ATP competitive small molecules targeting the CK2 α/β interface
16. Finding New Components of the Target of Rapamycin (TOR) Signaling Network through Chemical Genetics and Proteome Chips
17. Tryptophan in Multicomponent Petasis Reactions for Peptide Stapling and Late‐Stage Functionalisation
18. A fragment-based approach leading to the discovery of a novel binding site and the selective CK2 inhibitor CAM4066
19. A recombinant approach for stapled peptide discovery yields inhibitors of the RAD51 recombinase.
20. Studies Towards the Synthesis of the Core of Endiandric Acid H
21. Selective inhibitors of the Aurora A-TPX2 protein-protein interaction exhibit in vivo efficacy as targeted anti-mitotic agents
22. Studies on the biomimetic synthesis of the manzamine alkaloids
23. An expedient strategy for the diversity-oriented synthesis of macrocyclic compounds with natural product-like characteristics
24. Hybrid Androgen Receptor Inhibitors Outperform Enzalutamide and EPI‐001 in in vitro Models of Prostate Cancer Drug Resistance
25. Chapter 2. The Application of Diversity-oriented Synthesis in Chemical Biology
26. A cryptic hydrophobic pocket in the polo-box domain of the polo-like kinase PLK1 regulates substrate recognition and mitotic chromosome segregation
27. A cell-active cyclic peptide targeting the Nrf2/Keap1 protein–protein interaction.
28. A Recombinant Approach For Stapled Peptide Discovery Yields Inhibitors of the RAD51 Recombinase
29. The human proton pump inhibitors inhibit Mycobacterium tuberculosis rifampicin efflux and macrophage-induced rifampicin tolerance
30. Front Cover: Hybrid Androgen Receptor Inhibitors Outperform Enzalutamide and EPI‐001 in in vitro Models of Prostate Cancer Drug Resistance (ChemMedChem 2/2023)
31. Identification of macrocyclic peptides which activate bacterial cylindrical proteases
32. Synthesis of sp3-rich heterocyclic frameworks by a divergent synthesis strategy
33. Peroxide-cleavable linkers for antibody–drug conjugates
34. Disulfide re-bridging reagents for single-payload antibody-drug conjugates
35. A cell-active peptide targeting the Nrf2/Keap1 protein-protein interaction
36. Divergent and concise total syntheses of dihydrochalcones and 5-deoxyflavones recently isolated from Tacca species and Mimosa diplotricha
37. Overcoming Chemical, Biological, and Computational Challenges in the Development of Inhibitors Targeting Protein-Protein Interactions
38. Studies towards the synthesis of indolizin-5(3H)-one derivatives and related 6,5-azabicyclic scaffolds by ring-closing metathesis
39. Multifunctional supramolecular polymer networks as next-generation consolidants for archaeological wood conservation
40. LGR5 targeting molecules as therapeutic agents for multiple cancer types
41. Divinylpyrimidine reagents generate antibody-drug conjugates with excellent in vivo efficacy and tolerability
42. Synthesis of sp3-rich heterocyclic frameworks by a divergent synthesis strategy.
43. Antiplasmodial and trypanocidal activity of violacein and deoxyviolacein produced from synthetic operons
44. Rapid and robust cysteine bioconjugation with vinylheteroarenes
45. All-in-one disulfide bridging enables the generation of antibody conjugates with modular cargo loading
46. A two-component 'double-click' approach to peptide stapling
47. Applications of small molecule activators and inhibitors of quorum sensing in Gram-negative bacteria
48. A unified in vitro to in vivo fluorescence lifetime screening platform yields amyloid β aggregation inhibitors
49. A quorum-sensing molecule acts as a morphogen controlling gas vesicle organelle biogenesis and adaptive flotation in an enterobacterium
50. Diversity-oriented synthesis of macrocyclic peptidomimetics
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