1,639 results on '"Schols, Dominique"'
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2. Natural carboxyterminal truncation of human CXCL10 attenuates glycosaminoglycan binding, CXCR3A signaling and lymphocyte chemotaxis, while retaining angiostatic activity
3. Systematic assessment of chemokine ligand bias at the human chemokine receptor CXCR2 indicates G protein bias over β-arrestin recruitment and receptor internalization
4. Systemic cytokines and GlycA discriminate disease status and predict corticosteroid response in HTLV-1-associated neuroinflammation.
5. Steroidal 21-imidazolium salt derivatives: Synthesis and anticancer activity
6. Synthesis, molecular docking, dynamics study and preliminary cytotoxicity study of some coumarin linked imidazothiadiazoles
7. Design, synthesis, molecular docking, dynamics simulations and antiviral activities of quinoline derivatives
8. Synthesis of 3-heteroaryl-pyrrolo[2,3-b]pyridines as potent inhibitors of AP-2-associated protein kinase 1 (AAK1) with antiviral activity
9. Development of a cellular model to study CCR8 signaling in tumor-infiltrating regulatory T cells
10. Second generation Al18F-labeled D-amino acid peptide for CXCR4 targeted molecular imaging
11. Identification of novel human CC chemokine receptor 8 (CCR8) antagonists via the synthesis of naphthalene amide and sulfonamide isosteres
12. Synthesis and cancer cell cytotoxicity of 2-heteroaryl-4-(4-heteroaryl-2-oxobut-3-en-1-ylidene)-substituted benzothiazepanes
13. Synthesis and antitumor activity of cyclopentane-fused anthraquinone derivatives
14. Membrane-permeable tenofovir-di- and monophosphate analogues
15. Exploring antiviral potency of N-1 substituted pyrimidines against HIV-1 and other DNA/RNA viruses: Design, synthesis, characterization, ADMET analysis, docking, molecular dynamics and biological activity
16. Synthesis and structure–activity relationship study of phenoxybenzylpiperazine analogues as CCR8 agonists
17. PRO-2000 exhibits SARS-CoV-2 antiviral activity by interfering with spike-heparin binding
18. Synthesis of novel thioalkylated triazolothiazoles and their promising in-vitro antiviral activity
19. Cellular electrical impedance to profile SARS-CoV-2 fusion inhibitors and to assess the fusogenic potential of spike mutants
20. Anthranilamides with quinoline and β-carboline scaffolds: design, synthesis, and biological activity
21. Discovery of ( ±)-3-(1H-pyrazol-1-yl)-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4] thiadiazine derivatives with promising in vitro anticoronavirus and antitumoral activity
22. A stabilized CXCL9(74–103)-derived peptide selectively inhibits proliferation, adhesion and metastasis of tumor cells that express high levels of heparan sulfate
23. Potent neutralizing anti-SARS-CoV-2 human antibodies cure infection with SARS-CoV-2 variants in hamster model
24. Organotropic dendrons with high potency as HIV-1, HIV-2 and EV-A71 cell entry inhibitors
25. In silico design, synthesis and anti-HIV activity of quinoline derivatives as non-nucleoside reverse transcriptase inhibitors (NNRTIs)
26. Identification of novel chemotypes as CXCR2 antagonists via a scaffold hopping approach from a thiazolo[4,5-d]pyrimidine
27. Synthesis, in vitro cytotoxicity, molecular docking and ADME study of some indolin-2-one linked 1,2,3-triazole derivatives
28. Synthesis and evaluation of isothiazolo[4,5-b]pyridines as cyclin G-associated kinase (GAK) inhibitors.
29. Itaconic acid hybrids as potential anticancer agents
30. Exploring the dNTP -binding site of HIV-1 reverse transcriptase for inhibitor design
31. The nature of chronic rejection after lung transplantation: a murine orthotopic lung transplant study
32. Systematic Assessment of Human CCR7 Signalling Using NanoBRET Biosensors Points towards the Importance of the Cellular Context
33. Thiophene-2-carboxamide derivatives of anthraquinone: A new potent antitumor chemotype
34. Synthesis, molecular docking, and preliminary cytotoxicity study of some novel 2-(naphthalen-1-yl)-methylimidazo[2,1-b][1,3,4]thiadiazoles
35. Stimulation of the atypical chemokine receptor 3 (ACKR3) by a small-molecule agonist attenuates fibrosis in a preclinical liver but not lung injury model
36. Discovery of 3-phenyl- and 3-N-piperidinyl-isothiazolo[4,3-b]pyridines as highly potent inhibitors of cyclin G-associated kinase
37. Palladium-catalyzed cross-coupling reactions on a bromo-naphthalene scaffold in the search for novel human CC chemokine receptor 8 (CCR8) antagonists
38. Synthesis, in silico ADME, molecular docking and in vitro cytotoxicity evaluation of stilbene linked 1,2,3-triazoles
39. Alkylated benzimidazoles: Design, synthesis, docking, DFT analysis, ADMET property, molecular dynamics and activity against HIV and YFV
40. Radiosynthesis and preclinical evaluation of a 68Ga-labeled tetrahydroisoquinoline-based ligand for PET imaging of C-X-C chemokine receptor type 4 in an animal model of glioblastoma.
41. Rigid Macrocycle Metal Complexes as CXCR4 Chemokine Receptor Antagonists: Influence of Ring Size.
42. The Role of TIM-1 and CD300a in Zika Virus Infection Investigated with Cell-Based Electrical Impedance.
43. IL-10 predicts incident neuroinflammatory disease and proviral load dynamics in a large Brazilian cohort of people living with human T-lymphotropic virus type 1.
44. Synthesis and evaluation of sulfonamide derivatives of quinoxaline 1,4-dioxides as carbonic anhydrase inhibitors.
45. Amides of pyrrole- and thiophene-fused anthraquinone derivatives: A role of the heterocyclic core in antitumor properties
46. Design, Docking, Molecular Dynamics Simulations, Synthesis and Antiviral Activities of Quinoline Derivatives
47. Selective synthesis of an elusive C-functional bis-cyclam and study of its inhibition of the CXCR4 chemokine receptor
48. Trans-IV restriction: a new configuration for metal bis-cyclam complexes as potent CXCR4 inhibitors
49. A single-dose live-attenuated YF17D-vectored SARS-CoV-2 vaccine candidate
50. Potent Anti‐HIV Activity of Alkyl‐Modified DiPPro‐Nucleotides
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