170 results on '"Roman, David L."'
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2. High-Throughput GPCRome Screen of Pollutants Reveals the Activity of Polychlorinated Biphenyls at Melatonin and Sphingosine-1-phosphate Receptors
3. The Concise Guide to PHARMACOLOGY 2023/24: Introduction and Other Protein Targets
4. Screen Targeting Lung and Prostate Cancer Oncogene Identifies Novel Inhibitors of RGS17 and Problematic Chemical Substructures
5. Protein-protein interaction-based high throughput screening for adenylyl cyclase 1 inhibitors: Design, implementation, and discovery of a novel chemotype
6. Regulator of G Protein Signaling 17 as a Negative Modulator of GPCR Signaling in Multiple Human Cancers
7. Protein-Protein Interaction-Based High Throughput Screening For Adenylyl Cyclase 1 Inhibitors: Design, Implementation, and Discovery of a Novel Chemotype
8. Development of a Novel High-Throughput Screen and Identification of Small-Molecule Inhibitors of the Gα–RGS17 Protein–Protein Interaction Using AlphaScreen
9. THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Introduction and Other Protein Targets
10. New functional activity of aripiprazole revealed: Robust antagonism of D2 dopamine receptor-stimulated Gβγ signaling
11. Polyplexed Flow Cytometry Protein Interaction Assay: A Novel High-Throughput Screening Paradigm for RGS Protein Inhibitors
12. Regulators of G protein Signaling (RGS) proteins in GtoPdb v.2021.2
13. In vitro protein kinase activity measurement by flow cytometry
14. Microfabricated channel array electrophoresis for characterization and screening of enzymes using RGS-G protein interactions as a model system
15. Fragment‐Based Nuclear Magnetic Resonance Screen against a Regulator of G Protein Signaling Identifies a Binding “Hot Spot”
16. RGS17: an emerging therapeutic target for lung and prostate cancers
17. Chapter 11 Identification of Ligands Targeting RGS Proteins
18. Regulators of G protein Signaling (RGS) proteins (version 2020.5) in the IUPHAR/BPS Guide to Pharmacology Database
19. Regulator of G-protein signaling (RGS) proteins as drug targets: Progress and future potentials
20. Differential modulation of mu-opioid receptor signaling to adenylyl cyclase by regulators of G protein signaling proteins 4 or 8 and 7 in permeabilised C6 cells is Gα subtype dependent
21. Novel Peptide Ligands of RGS4 from a Focused One-Bead, One-Compound Library
22. Mechanism of Action and Structural Requirements of Constrained Peptide Inhibitors of RGS Proteins
23. Interactions of antidepressants with the serotonin transporter: a contemporary molecular analysis
24. Regulators of G protein Signaling (RGS) proteins (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database
25. High-resolution structure of RGS17 suggests a role for Ca2+ in promoting the GTPase-activating protein activity by RZ subfamily members
26. Evaluation of the Selectivity and Cysteine Dependence of Inhibitors across the Regulator of G Protein–Signaling Family
27. Identification of FDA-Approved Small Molecules Capable of Disrupting the Calmodulin–Adenylyl Cyclase 8 Interaction through Direct Binding to Calmodulin
28. Natural Products Discovered in a High-Throughput Screen Identified as Inhibitors of RGS17 and as Cytostatic and Cytotoxic Agents for Lung and Prostate Cancer Cell Lines
29. Development of a bimolecular luminescence complementation assay for RGS: G protein interactions in cells
30. Using NMR‐Based Fragment Screening to Probe the Druggability of Regulator of G Protein Signaling 17
31. Regulators of G protein signaling (RGS) Proteins as Drug Targets: Modulating GPCR Signal Transduction
32. Bias Analyses of Preclinical and Clinical D2 Dopamine Ligands: Studies with Immediate and Complex Signaling Pathways
33. Differential modulation of mu-opioid receptor signaling to adenylyl cyclase by RGS proteins 4 or 8 and 7 in permeabilised C6 cells is Gα subtype dependent
34. Evaluation of the Selectivity and Cysteine Dependence of Inhibitors across the Regulator of G Protein–Signaling Family
35. RABL6A, a Novel RAB-Like Protein, Controls Centrosome Amplification and Chromosome Instability in Primary Fibroblasts
36. Modification and Functional Inhibition of Regulator of G-Protein Signaling 4 (RGS4) by 4-Hydroxy-2-nonenal
37. A High Throughput Screen for RGS Proteins Using Steady State Monitoring of Free Phosphate Formation
38. TARGETING THE REGULATOR OF G PROTEIN SIGNALING 17 (RGS17) FOR LUNG AND PROSTATE CANCER TREATMENTS
39. Real-time monitoring of tyrosine hydroxylase activity using a plate reader assay
40. Expression and purification of recombinant human tyrosine hydroxylase as a fusion protein in Escherichia coli
41. Structural studies of RGS inhibitors
42. Book Review of Annual Review of Biochemistry. Volume 80
43. Regulators of G Protein Signaling (RGS) Proteins as Drug Targets: Modulating G-Protein-Coupled Receptor (GPCR) Signal Transduction
44. Book Review of Chemical Library Design
45. Book Review of Annual Review of Biochemistry. Volume 79
46. Reversible, Allosteric Small-Molecule Inhibitors of Regulator of G Protein Signaling Proteins
47. Allosteric Inhibition of the Regulator of G Protein Signaling–Gα Protein–Protein Interaction by CCG-4986
48. Use of Flow Cytometric Methods to Quantify Protein‐Protein Interactions
49. A covalent peptide inhibitor of RGS4 identified in a focused one-bead, one compound library screen
50. Assembly of High Order Gαq-Effector Complexes with RGS Proteins
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