25 results on '"Ohyama, Sumika"'
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2. The design and optimization of a series of 2-(pyridin-2-yl)-1 H-benzimidazole compounds as allosteric glucokinase activators
3. Structure–activity relationships of 3,5-disubstituted benzamides as glucokinase activators with potent in vivo efficacy
4. Discovery of potent and orally active 3-alkoxy-5-phenoxy- N-thiazolyl benzamides as novel allosteric glucokinase activators
5. Effect of long-term treatment with a small-molecule glucokinase activator on glucose metabolism, lipid profiles and hepatic function
6. Impact of Small-Molecule Glucokinase Activator on Glucose Metabolism and β-Cell Mass
7. Chronic sleep disorder induced by psychophysiological stress induces glucose intolerance without adipose inflammation in mice
8. Luminal dietary protein, not amino acids, induces pancreatic protease via CCK in pancreaticobiliary-diverted rats
9. Subgroup analysis of phase 3 studies of dulaglutide in Japanese patients with type 2 diabetes
10. Discovery of novel 2-(pyridine-2-yl)-1H-benzimidazole derivatives as potent glucokinase activators
11. Discovery and structure–activity relationships of a novel class of quinazoline glucokinase activators
12. Discovery of novel 3,6-disubstituted 2-pyridinecarboxamide derivatives as GK activators
13. Identification of novel and potent 2-amino benzamide derivatives as allosteric glucokinase activators
14. Continuous Exposure to a Novel Stressor Based on Water Aversion Induces Abnormal Circadian Locomotor Rhythms and Sleep-Wake Cycles in Mice
15. Pharmacokinetic and Pharmacodynamic Properties of the Glucokinase Activator MK-0941 in Rodent Models of Type 2 Diabetes and Healthy Dogs
16. Development and characterization of mouse model for stress induced sleep disorder
17. L-homoarginine suppresses exocrine pancreas in rats.
18. The design and optimization of a series of 2-(pyridin-2-yl)-1H-benzimidazole compounds as allosteric glucokinase activators
19. A selective small molecule glucagon-like peptide-1 secretagogue acting via depolarization-coupled Ca2+ influx
20. Impact of Small-Molecule Glucokinase Activator on Glucose Metabolism and β-Cell Mass
21. Metabolic impact of overexpression of liver glycogen synthase with serine-to-alanine substitutions in rat primary hepatocytes
22. An Allosteric Activator of Glucokinase Impairs the Interaction of Glucokinase and Glucokinase Regulatory Protein and Regulates Glucose Metabolism
23. Endogenous cholecystokinin plays a role in down-regulation of pancreatic amylase independent of dietary carbohydrate in rats
24. Impact of Small Molecule Glucokinase Activator on Glucose Metabolism in Response to High-Fat-Diet in Mice with β-Cell Specific Haploinsufficiency of Glucokinase Gene.
25. Impact of small-molecule glucokinase activator on glucose metabolism and beta-cell mass.
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