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This paper highlights qualitatively and quantitatively research and presents a valuable overview of new citation enhanced databases in the context of research evaluation for the productivity of Prof. Jayant V. Narlikar. He has total 472 research publications in the fields of Astronomy and Astrophysics (AA) published from 1961-2015. In addition, this paper provides an overview of the citation-enhanced databases viz Astrophysics Data System Beta: A powerful new interface for performing citation analysis. Previously, scientometrics had been used to measure the publication productivity of Prof. Jayant V. Narlikar using the Astrophysics Data System (ADS). The scope of this paper is limited to Astrophysics Data System Beta. The result indicates that most of his papers are published in peer reviewed journals having the highest Impact Factor. The average number of publications per year is 8.74 and with the maximum papers published during 1981-1990 and 1996-2000. The total number of citations for his publications is 3516 covering 665 of his papers published during 1961-1970. He had many research collaborations, specifically with Prof. F. Hoyle (87 papers), Prof. G. Burbidge (38 papers), Prof. N. Wickramasinghe (22 papers) and Prof. T. Padmanabhan (21 papers).

An improved and rapid synthesis of mefenamic acid based indole derivatives has been achieved via the ligand free Cu-catalyzed coupling-cyclization method under ultrasound irradiation. This simple, straightforward and inexpensive one-pot method involved the reaction of a terminal alkyne derived from mefenamic acid with 2-iodosulfanilides in the presence of CuI and K 2 CO 3 in PEG-400. The reaction proceeded via an initial CC bond formation (the coupling step) followed by CN bond formation (the intramolecular cyclization) to afford the mefenamic acid based indole derivatives in good to acceptable yields. Several of these compounds showed inhibition of PDE4 in vitro and the SAR (Structure Activity Relationship) within the series is discussed. The compound 3d has been identified as a promising and selective inhibitor of PDE4B (IC 50  = 1.34 ± 0.46 µM) that showed TNF-α inhibition in vitro (IC 50  = 5.81 ± 0.24 µM) and acceptable stability in the rat liver microsomes., Competing Interests: Declaration of Competing Interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper., (Copyright © 2020 Elsevier Ltd. All rights reserved.)