175 results on '"Mosley, Ralph T."'
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2. Synthesis and Biological Activities of Potent Peptidomimetics Selective for Somatostatin Receptor Subtype 2
3. What's all the FLAP about?: 5-lipoxygenase-activating protein inhibitors for inflammatory diseases
4. Structure and chemistry of apicidins, a class of novel cyclic tetrapeptides without a terminal alpha-keto epoxide as inhibitors of histone deacetylase with potent antiprotozoal activities
5. Assignment of the liposidomycin diazepanone stereochemistry
6. Peptidomimetics
7. Synthesis nd biological activities of potent peptidomimetics selective for somatostatin receptor subtype 2
8. Structure–activity relationship of linear tetrapeptides Tic-DPhe-Arg-Trp-NH2 at the human melanocortin-4 receptor and effects on feeding behaviors in rat
9. Amino acid substitution of arginine 80 in 17β-hydroxysteroid dehydrogenase type 3 and its effect on NADPH cofactor binding and oxidation/reduction kinetics
10. A simple method for visualizing the differences between related receptor sites
11. Correction to Nucleoside, Nucleotide, and Non-Nucleoside Inhibitors of Hepatitis C Virus NS5B RNA-Dependent RNA-Polymerase
12. Inhibition of hepatitis C virus NS5A by fluoro-olefin based γ-turn mimetics
13. Phenylpropenamide derivatives: Anti-hepatitis B virus activity of the Z isomer, SAR and the search for novel analogs
14. Molecular and Structural Basis for the Roles of Hepatitis C Virus Polymerase NS5B Amino Acids 15, 223, and 321 in Viral Replication and Drug Resistance
15. Discovery of a Novel Class of Potent HCV NS4B Inhibitors: SAR Studies on Piperazinone Derivatives
16. Use of 2′-Spirocyclic Ethers in HCV Nucleoside Design
17. The synthesis and conformational analysis of amino acid–tetrahydroanthranilic acid hybrids
18. Structure of Hepatitis C Virus Polymerase in Complex with Primer-Template RNA
19. Nucleoside, Nucleotide, and Non-Nucleoside Inhibitors of Hepatitis C Virus NS5B RNA-Dependent RNA-Polymerase
20. Benzimidazolones: A New Class of Selective Peroxisome Proliferator-Activated Receptor γ (PPARγ) Modulators
21. Adenosine Deaminase-like Protein 1 (ADAL1): Characterization and Substrate Specificity in the Hydrolysis of N6- or O6-Substituted Purine or 2-Aminopurine Nucleoside Monophosphates
22. Benzo[b]thiophene-based histone deacetylase inhibitors
23. Androstene-3,5-dienes as ER-β selective SERMs
24. The discovery of 6-amino nicotinamides as potent and selective histone deacetylase inhibitors
25. Novel glucocorticoids containing a 6,5-bicyclic core fused to a pyrazole ring: Synthesis, in vitro profile, molecular modeling studies, and in vivo experiments
26. Estrogen receptor ligands. Part 16: 2-Aryl indoles as highly subtype selective ligands for ERα
27. Identification of small molecule estrogen-related receptor α-specific antagonists and homology modeling to predict the molecular determinants as the basis for selectivity over ERRβ and ERRγ
28. The Differential Interactions of Peroxisome Proliferator-Activated Receptor γ Ligands with Tyr473 Is a Physical Basis for Their Unique Biological Activities
29. Sordarin Derivatives Induce a Novel Conformation of the Yeast Ribosome Translocation Factor eEF2
30. Tetrahydrofluorenones with conformationally restricted side chains as selective estrogen receptor beta ligands
31. Androstenediol analogs as ER-β-selective SERMs
32. Estrogen receptor ligands. Part 14: Application of novel antagonist side chains to existing platforms
33. Reagent Selector: Using Synthon Analysis to Visualize Reagent Properties and Assist in Combinatorial Library Design.
34. Estrogen receptor ligands. Part 11: Synthesis and activity of isochromans and isothiochromans
35. Selective glucocorticoid receptor nonsteroidal ligands completely antagonize the dexamethasone mediated induction of enzymes involved in gluconeogenesis and glutamine metabolism
36. Comparison of 2‐Phenylspiroindenes and 2‐Phenylspiroindenediones as Estrogen Receptor Ligands — Modeling and Binding Data Don′t Agree!
37. Estrogen Receptor Ligands. II. Discovery of Benzoxathiins as Potent, Selective Estrogen Receptor α Modulators
38. Estrogen receptor ligands. Part 1: The discovery of flavanoids with subtype selectivity
39. Comparison of 2-phenylspiroindenes and 2-phenylspiroindenediones as estrogen receptor ligands—modeling and binding data don't agree!
40. 2-Phenylspiroindenes: A Novel Class of Selective Estrogen Receptor Modulators (SERMs).
41. 1H-NMR studies on a potent and selective antagonist at human melanocortin receptor 4 (hMC-4R)
42. 2-Phenylspiroindenes: a novel class of selective estrogen receptor modulators (SERMs)
43. Erratum to “A simple method for visualizing the differences between related receptor sites”
44. Combinatorial library of indinavir analogues: replacement for the aminoindanol at P2′
45. Design and Pharmacology of N-[(3R)-1,2,3,4-Tetrahydroisoquinolinium- 3-ylcarbonyl]-(1R)-1-(4-chlorobenzyl)- 2-[4-cyclohexyl-4-(1H-1,2,4-triazol- 1-ylmethyl)piperidin-1-yl]-2-oxoethylamine (1), a Potent, Selective, Melanocortin Subtype-4 Receptor Agonist
46. Structure and Chemistry of Apicidins, a Class of Novel Cyclic Tetrapeptides without a Terminal α-Keto Epoxide as Inhibitors of Histone Deacetylase with Potent Antiprotozoal Activities
47. ChemInform Abstract: Assignment of the Liposidomycin Diazepanone Stereochemistry.
48. Use of 2′-SpirocyclicEthers in HCV NucleosideDesign.
49. Discovery of a Novel Classof Potent HCV NS4B Inhibitors:SAR Studies on Piperazinone Derivatives.
50. A Combinatorial Approach toward the Discovery of Non-Peptide, Subtype-Selective Somatostatin Receptor Ligands
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