677 results on '"Marinelli, Luciana"'
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2. A reverse translational approach reveals the protective roles of Mangifera indica in inflammatory bowel disease
3. Exploring the 1,3-benzoxazine chemotype for cannabinoid receptor 2 as a promising anti-cancer therapeutic
4. Theoretical and experimental studies on the interaction of biphenyl ligands with human and murine PD-L1: Up-to-date clues for drug design
5. Discovery of 2,3-Diaminoindole Derivatives as a Novel Class of NOD Antagonists
6. The organometallic ferrocene exhibits amplified anti-tumor activity by targeted delivery via highly selective ligands to αvβ3, αvβ6, or α5β1 integrins
7. Design, synthesis and biological evaluation of novel TRβ selective agonists sustained by ADME-toxicity analysis
8. A combined approach of structure‐based virtual screening and NMR to interrupt the PD‐1/PD‐L1 axis: Biphenyl‐benzimidazole containing compounds as novel PD‐L1 inhibitors
9. Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases
10. A combined approach of structure‐based virtual screening and NMR to interrupt the PD‐1/PD‐L1 axis: Biphenyl‐benzimidazole containing compounds as novel PD‐L1 inhibitors.
11. Development and Nanoparticle-Mediated Delivery of Novel MDM2/MDM4 Heterodimer Peptide Inhibitors to Enhance 5‑Fluorouracil Nucleolar Stress in Colorectal Cancer Cells.
12. Molecular View on the iRGD Peptide Binding Mechanism: Implications for Integrin Activity and Selectivity Profiles
13. Minute-timescale simulations of G Protein Coupled Receptor A2A activation mechanism reveals a receptor pseudo-active state
14. Cationic nucleopeptides as novel non-covalent carriers for the delivery of peptide nucleic acid (PNA) and RNA oligomers
15. Challenging clinically unresponsive medullary thyroid cancer: Discovery and pharmacological activity of novel RET inhibitors
16. Isocyanides as Catalytic Electron Acceptors in the Visible Light Promoted Oxidative Formation of Benzyl and Acyl Radicals
17. Retromer stabilization results in neuroprotection in a model of Amyotrophic Lateral Sclerosis
18. HuR modulation counteracts lipopolysaccharide response in murine macrophages
19. Locking PDK1 in DFG-out conformation through 2-oxo-indole containing molecules: Another tools to fight glioblastoma
20. Chemical modifications in the seed region of miRNAs 221/222 increase the silencing performances in gastrointestinal stromal tumor cells
21. Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation
22. Molecular View on the iRGD Peptide Binding Mechanism: Implications for Integrin Activity and Selectivity Profiles.
23. HuR modulation with tanshinone mimics impairs LPS response in murine macrophages
24. Tanshinone Mimics Bearing a 3-Heterocyclic Ring Endowed with Increased Solubility and Anti-Inflammatory Properties
25. Synthesis, biological activity and molecular modeling of new biphenylic carboxamides as potent and selective CB2 receptor ligands
26. Identification of a Novel p53 Modulator Endowed with Antitumoural and Antibacterial Activity through a Scaffold Repurposing Approach
27. A Small CEACAM5 Peptide Restores the Protective Function of CD8+ Regulatory T Cells in Crohn’s Disease
28. A stereoselective approach to peptidomimetic BACE1 inhibitors
29. Pharmacological folding chaperones act as allosteric ligands of Frizzled4
30. Sampling protein motion and solvent effect during ligand binding
31. Progresses in the pursuit of aldose reductase inhibitors: The structure-based lead optimization step
32. Identification of novel molecular scaffolds for the design of MMP-13 inhibitors: A first round of lead optimization
33. HuR-targeted agents: An insight into medicinal chemistry, biophysical, computational studies and pharmacological effects on cancer models
34. Molecular basis of cyclooxygenase enzymes (COXs) selective inhibition
35. Identification of 5-arylidene-4-thiazolidinone derivatives endowed with dual activity as aldose reductase inhibitors and antioxidant agents for the treatment of diabetic complications
36. Synthesis and biological evaluation in U87MG glioma cells of (ethynylthiophene)sulfonamido-based hydroxamates as matrix metalloproteinase inhibitors
37. Temozolomide-Acquired Resistance Is Associated with Modulation of the Integrin Repertoire in Glioblastoma, Impact of α5β1 Integrin
38. Enriching the Arsenal of Pharmacological Tools against MICAL2
39. Site-directed Mutagenesis of Key Residues Unveiled a Novel Allosteric Site on Human Adenosine Kinase for Pyrrolobenzoxa(thia)zepinone Non-Nucleoside Inhibitors
40. Interfering with the Tumor–Immune Interface: Making Way for Triazine-Based Small Molecules as Novel PD-L1 Inhibitors
41. Halting the Spread of Herpes Simplex Virus-1: The Discovery of an Effective Dual αvβ6/αvβ8 Integrin Ligand
42. Highly Selective Cyclic Hexapeptides Antagonist of GPIIb-IIIa by Multiple N-Methylation
43. Novel Peptide-Based PET Probe for Non-invasive Imaging of C-X-C Chemokine Receptor Type 4 (CXCR4) in Tumors
44. Click-Chemistry (CuAAC) Trimerization of an αvβ₆ Integrin Targeting Ga-68-Peptide : Enhanced Contrast for in-Vivo PET Imaging of Human Lung Adenocarcinoma Xenografts
45. Human recombinant beta-secretase immobilized enzyme reactor for fast hits’ selection and characterization from a virtual screening library
46. Conformational analysis of furanoid [member of]-sugar amino acid containing cyclic peptides by NMR spectroscopy, molecular dynamics simulation, and X-ray crystallography: Evidence for a novel turn structure
47. N-O-Isopropyl sulfonamido-based hydroxamates: Kinetic characterisation of a series of MMP-12/MMP-13 dual target inhibitors
48. Disulfide Bond Replacement with 1,4‐ and 1,5‐Disubstituted [1,2,3]‐Triazole on C‐X‐C Chemokine Receptor Type 4 (CXCR4) Peptide Ligands: Small Changes that Make Big Differences
49. Click‐Chemistry (CuAAC) Trimerization of an αvβ6 Integrin Targeting Ga‐68‐Peptide: Enhanced Contrast for in‐Vivo PET Imaging of Human Lung Adenocarcinoma Xenografts
50. Targeting the KRAS oncogene: Synthesis, physicochemical and biological evaluation of novel G-Quadruplex DNA binders
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