299 results on '"Makhaeva G"'
Search Results
2. Influence of the sulfonyl group on the biological activity of 2-sulfonarylhydrazinylidene 1,3-dicarbonyl compounds
3. Synthesis of conjugates of ipidacrine with oxa/azaheterocycles and their potential as agents for the treatment of Alzheimer’s disease
4. Conjugates of tacrine with aminomethylidene derivatives of ethyl acetoacetate as promising agents for the treatment of Alzheimer’s disease
5. Multifunctional Inhibitors of Cholinesterases for the Therapy of Alzheimer’s Disease (A Review)
6. New highly efficient multifunctional cholinesterase inhibitors based on the conjugation of amiridine and tacrine homolog
7. Amino Derivatives of Acridine: Synthesis and Study of Anticholinesterase and Antioxidant Activity
8. Synthesis and properties of new derivatives of 4-amino-2,3-polymethylenequinolines with antioxidant function
9. Multipharmacophore strategy in medicinal chemistry for the design of drugs for the treatment of Alzheimer’s and some other neurodegenerative diseases
10. Synthesis and study of the biological activity of thiourea-containing amiridine derivatives as potential multi-target drugs for the treatment of Alzheimer’s disease
11. Conjugates of Tacrine with Aminomethylidene-Substituted Malonates: Synthesis and Biological Evaluation
12. Tacrine Derivatives Containing an Antioxidant Moiety
13. 3-(2-Arylhydrazono)-1,1,1-trifluro-3-(phenylsulfonyl)propan-2-ones as selective carboxylesterase inhibitors
14. Synthesis of new efficient and selective carboxylesterase inhibitors based on adamantyl and citronellyl 4,4,4-trifluoro-2-arylhydrazonylidene-3-oxobutanoates
15. Neuroprotective and Antioxidant Activity of Arachidonoyl Choline, Its Bis-Quaternized Analogues and Other Acylcholines
16. Cholinesterase and carboxylesterase inhibitors as pharmacological agents
17. Anticholinesterase and Antioxidant Activity of New Binary Conjugates of γ-Carbolines
18. Synthesis and biological activity of 5-vinyl- and 5-allyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indoles
19. Aminoadamantane conjugates with carbazole derivatives as potential multitarget agents for the treatment of Alzheimer’s disease. Effect of the spacer structure
20. Influence of the γ-carboline and carbazole pharmacophore moieties on anticholinesterase and antiradical activity of multifunctional agents for the treatment of neurodegenerative diseases
21. AMINO DERIVATIVES OF ACRIDINE: SYNTHESIS, STUDY OF ANTICHOLINESTERASE AND ANTIOXIDANT ACTIVITIES
22. Synthesis of γ-carbolines containing NO-donor fragment and assessment of their anticholinesterase activity
23. Multi-Strip Assay and Multimodal Biosensors for Environmental and Medical Monitoring of Neurotoxicants
24. Blood Esterases as a Complex Biomarker for Exposure to Organophosphorus Compounds
25. Chemical Similarity, Shape Matching and QSAR
26. Molecular polymorphism of human enzymes as the basis of individual sensitivity to drugs. Supercomputer-assisted modeling as a tool for analysis of structural changes and enzymatic activity of proteins
27. 1,2,4-Thiadiazoles as promising multifunctional agents for treatment of neurodegenerative diseases
28. Synthesis and studies of biological activity of N-(4-tert-butylbenzyl)-N-(pyridin-3-ylmethyl)-2-aminothiazolines as potential multifunctional agents for treatment of neurodegenerative diseases
29. Molecular design of N,N-disubstituted 2-aminothiazolines as selective carboxylesterase inhibitors
30. Alkyl 2-arylhydrazinylidene-3-oxo-3-polyfluoroalkylpropionates as new effective and selective inhibitors of carboxylesterase
31. Esterase profiles of hexafluoropropan-2-ol-based dialkyl phosphates as a major determinant of their effects in mouse brain in vivo
32. Synthesis and investigation of biological activity of phosphorylated amines and amides
33. Kinetics and mechanism of inhibition of serine esterases by fluorinated carbethoxy 1-aminophosphonates
34. Synthesis and biological activity of O-carbamoylated 1,1,1,3,3,3-hexafluoroisopropanols as new specific inhibitors of carboxylesterase
35. Esterase profile of O-phosphorylated ethyltrifluorolactates in prediction of their therapeutic and toxic effects
36. Molecular design of O-phosphorylated oximes—Selective inhibitors of butyrylcholinesterase
37. Synthesis of O-phosphorylated 1-substituted 2,2,2-trifluoroethanols, serine hydrolase inhibitors
38. Study of the structural determinants of acute and delayed neurotoxicity of O-phosphorylated oximes by molecular field topology analysis (MFTA)
39. Esterase profile and analysis of structure-inhibitor selectivity relationships for homologous phosphorylated 1-hydroperfluoroisopropanols
40. Modeling of the relationships between the structure of O-phosphorylated oximes and their anticholinesterase activity and selectivity using molecular field topology analysis (MFTA)
41. Fluorinated α-aminophosphonates—a new type of irreversible inhibitors of serine hydrolases
42. N,N-disubstituted 2-aminothiazolines as new inhibitors of serine esterases
43. A new selective inhibitor of mouse blood plasma carboxylesterase
44. NTE and neuropathies induced by OP compounds: SW02.W9–6
45. Assessment of the Neurotoxic Potential of Some Methyl- and Phenylphosphonates Using a Stable Preparation of Neuropathy Target Esterase from Chicken Brain
46. Multi-Strip Assay and Multimodal Biosensors for Environmental and Medical Monitoring of Neurotoxicants
47. Blood Esterases as a Complex Biomarker for Exposure to Organophosphorus Compounds
48. Comparative Analysis of Esterase Activities of Human, Mouse, and Rat Blood
49. Dialkyl (1-ethoxycarbonyl-2,2,2-trifluoro-1-phenylsulfonylaminoethyl)-phosphonates
50. Study of the relationship between spatial structure and anticholinesterase activity of o-phosphorylate oximes
Catalog
Books, media, physical & digital resources
Discovery Service for Jio Institute Digital Library
For full access to our library's resources, please sign in.