330 results on '"Majumdar, Susruta"'
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2. Oxa-Iboga alkaloids lack cardiac risk and disrupt opioid use in animal models
3. Design and structural validation of peptide–drug conjugate ligands of the kappa-opioid receptor
4. Ligand and G-protein selectivity in the κ-opioid receptor
5. Insights into distinct signaling profiles of the µOR activated by diverse agonists
6. IUPHAR themed review: Opioid efficacy, bias, and selectivity
7. Structure-based design of bitopic ligands for the µ-opioid receptor
8. Agonist-selective recruitment of engineered protein probes and of GRK2 by opioid receptors in living cells.
9. Opioid signaling and design of analgesics
10. Machine Learning Harnesses Molecular Dynamics to Discover New $\mu$ Opioid Chemotypes
11. Canvass: A Crowd-Sourced, Natural-Product Screening Library for Exploring Biological Space.
12. The Functional Diversity of G Proteins in Opioid Receptor Signaling
13. Efficacy modulation by targeting the sodium binding allosteric site in the delta opioid receptor
14. Structural Analysis of Delta Opioid Receptor Ligands for Chronic Pain Therapeutics
15. Kratom Alkaloids, Natural and Semi-Synthetic, Show Less Physical Dependence and Ameliorate Opioid Withdrawal
16. Synthesis and Characterization of Azido Aryl Analogs of IBNtxA for Radio-Photoaffinity Labeling Opioid Receptors in Cell Lines and in Mouse Brain
17. Signaling Modulation Mediated by Ligand Water Interactions with the Sodium Site at μOR.
18. Site selective C–H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy
19. Imaging Sigma-1 Receptor (S1R) Expression Using Iodine-124-Labeled 1-(4-Iodophenyl)-3-(2-adamantyl)guanidine ([124I]IPAG)
20. Synthesis of spiro-2,6-dioxopiperazine and spiro-2,6-dioxopyrazine scaffolds using amino acids in a three-component reaction to generate potential Sigma-1 (σ1) receptor selective ligands
21. Negative allosteric modulation of the µ-opioid receptor
22. The antinociceptive effects of a dual kappa-delta opioid receptor agonist in the mouse formalin test
23. Structure, Function, and Pharmacology of Delta Opioid Receptor Bitopics
24. Structure based approaches on fentanyl template to design novel mu opioid modulators
25. Truncated mu opioid GPCR variant involvement in opioid-dependent and opioid-independent pain modulatory systems within the CNS
26. Pharmacological Characterization of Levorphanol, a G-Protein Biased Opioid Analgesic
27. Strategy for making safer opioids bolstered
28. Genetic dissociation of morphine analgesia from hyperalgesia in mice
29. Structure-based design of bitopic ligands for the µ-opioid receptor
30. Insights into distinct signaling profiles of the µOR activated by diverse agonists
31. Broad-spectrum analgesic efficacy of IBNtxA is mediated by exon 11-associated splice variants of the mu-opioid receptor gene
32. Truncated μ-Opioid Receptors With 6 Transmembrane Domains Are Essential for Opioid Analgesia
33. Isocyanide-Based Multicomponent Reactions Based upon Intramolecular Nitrilium Trapping
34. Strategies towards safer opioid analgesics—A review of old and upcoming targets.
35. Truncated G protein-coupled mu opioid receptor MOR-1 splice variants are targets for highly potent opioid analgesics lacking side effects
36. The mixed kappa and delta opioid receptor agonist, MP1104, attenuates chemotherapy-induced neuropathic pain
37. Strategies towards safer opioid analgesics—A review of old and upcoming targets
38. Structural insights into distinct signaling profiles of the μOR activated by diverse agonists
39. Radioligand Binding Assay for an Exon 11-Associated Mu Opioid Receptor Target
40. Oxidative Metabolism as a Modulator of Kratom’s Biological Actions
41. Evaluation of Kratom Opioid Derivatives as Potential Treatment Option for Alcohol Use Disorder
42. Alternative Pre-mRNA Splicing of the Mu Opioid Receptor Gene, OPRM1: Insight into Complex Mu Opioid Actions
43. A Novel Mitragynine Analog with Low-Efficacy Mu Opioid Receptor Agonism Displays Antinociception with Attenuated Adverse Effects
44. Mediation of opioid analgesia by a truncated 6-transmembrane GPCR
45. Novel Class of Psychedelic Iboga Alkaloids Disrupts Opioid Addiction States
46. Kratom Alkaloids as Probes for Opioid Receptor Function: Pharmacological Characterization of Minor Indole and Oxindole Alkaloids from Kratom
47. Prodrugs of Theophylline Incorporating Ethyleneoxy Groups in the Promoiety: Synthesis, Characterization, and Transdermal Delivery
48. The effect of water solubility of solutes on their flux through human skin in vitro: A prodrug database integrated into the extended Flynn database
49. An efficient 1,3-allylic carbonyl transposition of chalcones
50. Pharmacological Characterization of Synthetic Kratom Alkaloids for Improved Alcohol Use Disorder Therapeutics
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