22 results on '"Kosaka, Takatoshi"'
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2. trans-3,4-Disubstituted pyrrolidines as inhibitors of the human aspartyl protease renin. Part II: Prime site exploration using an oxygen linker
3. Identification of a Novel Allosteric Inhibitory Site on Tryptophan Hydroxylase 1 Enabling Unprecedented Selectivity Over all Related Hydroxylases
4. Novel ROCK inhibitors for the treatment of pulmonary arterial hypertension
5. trans -(3 S ,4 S )-Disubstituted pyrrolidines as inhibitors of the human aspartyl protease renin. Part I: Prime site exploration using an amino linker
6. Implementation of pharmacokinetic and pharmacodynamic strategies in early research phases of drug discovery and development at Novartis Institute of Biomedical Research
7. Structure-Based Design of Substituted Piperidines as a New Class of Highly Efficacious Oral Direct Renin Inhibitors
8. A Novel Class of Oral Direct Renin Inhibitors: Highly Potent 3,5-Disubstituted Piperidines Bearing a Tricyclic P3–P1 Pharmacophore
9. The Discovery of Novel Potent trans-3,4-Disubstituted Pyrrolidine Inhibitors of the Human Aspartic Protease Renin from in Silico Three-Dimensional (3D) Pharmacophore Searches
10. Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-Cyanopyrimidines. Part 2
11. 4-Amino-2-cyanopyrimidines: Novel scaffold for nonpeptidic cathepsin S inhibitors
12. Discovery of selective and nonpeptidic cathepsin S inhibitors
13. Discovery of Orally Bioavailable Cathepsin S Inhibitors for the Reversal of Neuropathic Pain
14. Effect of Cathepsin K Inhibitors on Bone Resorption
15. Remarkable Difference of Phase Transition Behaviors Between Langmuir Monolayers and Aqueous Bilayer Vesicles of Oligopeptide-Carrying Lipids
16. Studies on 5-Lipoxygenase Inhibitors. Synthesis of and Structure-Activity Relationship in p-Hydroxyarylalkenylbenzoazoles
17. Synthesis of Ethenylbenzothiazole Derivatives
18. Enantioselective synthesis of neoambrosin, parthenin, and dihydroisoparthenin
19. Synthesis of 2-(4-Aryl-1E,3E-butadienyl)benzoxazoles by the Horner-Wadsworth-Emmons Reaction
20. A novel series of highly potent 5-lipoxygenase inhibitors; 2-aryldienylbenzoxazoles
21. The Discoveryof Novel Potent trans-3,4-Disubstituted Pyrrolidine Inhibitors of the Human Aspartic Protease Renin from in Silico Three-Dimensional (3D) Pharmacophore Searches.
22. Total Synthesis of Clavukerin A and Its Epimer
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