1. Structure-Based Design and Pharmacokinetic Optimization of Covalent Allosteric Inhibitors of the Mutant GTPase KRASG12C
- Author
-
Kettle, Jason G., primary, Bagal, Sharan K., additional, Bickerton, Sue, additional, Bodnarchuk, Michael S., additional, Breed, Jason, additional, Carbajo, Rodrigo J., additional, Cassar, Doyle J., additional, Chakraborty, Atanu, additional, Cosulich, Sabina, additional, Cumming, Iain, additional, Davies, Michael, additional, Eatherton, Andrew, additional, Evans, Laura, additional, Feron, Lyman, additional, Fillery, Shaun, additional, Gleave, Emma S., additional, Goldberg, Frederick W., additional, Harlfinger, Stephanie, additional, Hanson, Lyndsey, additional, Howard, Martin, additional, Howells, Rachel, additional, Jackson, Anne, additional, Kemmitt, Paul, additional, Kingston, Jennifer K., additional, Lamont, Scott, additional, Lewis, Hilary J., additional, Li, Songlei, additional, Liu, Libin, additional, Ogg, Derek, additional, Phillips, Christopher, additional, Polanski, Radek, additional, Robb, Graeme, additional, Robinson, David, additional, Ross, Sarah, additional, Smith, James M., additional, Tonge, Michael, additional, Whiteley, Rebecca, additional, Yang, Junsheng, additional, Zhang, Longfei, additional, and Zhao, Xiliang, additional
- Published
- 2020
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