456 results on '"Hsieh, Hsing-Pang"'
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2. A dual nociceptin and mu opioid receptor agonist exhibited robust antinociceptive effect with decreased side effects
3. Design of drug-like hepsin inhibitors against prostate cancer and kidney stones
4. Targeting cathepsin S promotes activation of OLF1-BDNF/TrkB axis to enhance cognitive function
5. Novel FLT3/AURK multikinase inhibitor is efficacious against sorafenib-refractory and sorafenib-resistant hepatocellular carcinoma
6. A critical overview of current progress for COVID-19: development of vaccines, antiviral drugs, and therapeutic antibodies
7. Natural product myricetin is a pan-KDM4 inhibitor which with poly lactic-co-glycolic acid formulation effectively targets castration-resistant prostate cancer
8. Design and synthesis of novel orally selective and type II pan-TRK inhibitors to overcome mutations by property-driven optimization
9. Discovery of Dual MER/AXL Kinase Inhibitors as Bifunctional Small Molecules for Inhibiting Tumor Growth and Enhancing Tumor Immune Microenvironment.
10. Influence of Ring Strain on the Formation of Rearrangement vs Cyclization Isotwistane Products in the Acyl Radical Reaction of Bicyclo[2.2.2]octanone
11. Design and synthesis of BPR1K653 derivatives targeting the back pocket of Aurora kinases for selective isoform inhibition
12. Discovery of novel inhibitors of Aurora kinases with indazole scaffold: In silico fragment-based and knowledge-based drug design
13. Development of Furanopyrimidine-Based Orally Active Third-Generation EGFR Inhibitors for the Treatment of Non-Small Cell Lung Cancer
14. Dual Kit/Aur Inhibitors as Chemosensitizing Agents for the Treatment of Melanoma: Design, Synthesis, Docking Studies and Functional Investigation
15. Recent advances in total synthesis of natural products by masked ortho ‐benzoquinones
16. Ligand efficiency based approach for efficient virtual screening of compound libraries
17. Aurora kinase inhibitors reveal mechanisms of HURP in nucleation of centrosomal and kinetochore microtubules
18. Identification of ligand efficient, fragment-like hits from an HTS library: structure-based virtual screening and docking investigations of 2H- and 3H-pyrazolo tautomers for Aurora kinase A selectivity
19. Identification of Entry Inhibitors against Delta and Omicron Variants of SARS-CoV-2
20. Additional file 1 of A critical overview of current progress for COVID-19: development of vaccines, antiviral drugs, and therapeutic antibodies
21. Additional file 1 of Natural product myricetin is a pan-KDM4 inhibitor which with poly lactic-co-glycolic acid formulation effectively targets castration-resistant prostate cancer
22. Additional file 1 of Novel FLT3/AURK multikinase inhibitor is efficacious against sorafenib-refractory and sorafenib-resistant hepatocellular carcinoma
23. Additional file 3 of Novel FLT3/AURK multikinase inhibitor is efficacious against sorafenib-refractory and sorafenib-resistant hepatocellular carcinoma
24. Synthesis and biological evaluation of 1-(4′-Indolyl and 6′-Quinolinyl) indoles as a new class of potent anticancer agents
25. Discovery of BPR1R024, an Orally Active and Selective CSF1R Inhibitor that Exhibits Antitumor and Immunomodulatory Activity in a Murine Colon Tumor Model
26. Chlorinated briarane diterpenoids from octocoral Briareum stechei (Kükenthal, 1908)
27. Aurintricarboxylic acid inhibits influenza virus neuraminidase
28. BPR-3P0128 inhibits RNA-dependent RNA polymerase elongation and VPg uridylylation activities of Enterovirus 71
29. Colloidal Assemblies Composed of Polymeric Micellar/Emulsified Systems Integrate Cancer Therapy Combining a Tumor-Associated Antigen Vaccine and Chemotherapeutic Regimens
30. A cell-based high-throughput screen for epidermal growth factor receptor pathway inhibitors
31. Anti-HSV activity of digitoxin and its possible mechanisms
32. Reactions of 2-hydroxybenzophenones with Corey–Chaykovsky reagent
33. CDKN1A-mediated responsiveness of MLL-AF4-positive acute lymphoblastic leukemia to Aurora kinase-A inhibitors
34. Mimicking H3 Substrate Arginine in the Design of G9a Lysine Methyltransferase Inhibitors for Cancer Therapy: A Computational Study for Structure-Based Drug Design
35. Development of a Robust Scale-Up Synthetic Route for BPR1K871: A Clinical Candidate for the Treatment of Acute Myeloid Leukemia and Solid Tumors
36. Development and validation of a liquid chromatography–tandem mass spectrometry for the determination of BPR0L075, a novel antimicrotuble agent, in rat plasma: Application to a pharmacokinetic study
37. Isocostunolide, a sesquiterpene lactone, induces mitochondrial membrane depolarization and caspase-dependent apoptosis in human melanoma cells
38. Briarenols W–Z: Chlorine-Containing Polyoxygenated Briaranes from Octocoral Briareum stechei (Kükenthal, 1908)
39. One-Pot Synthesis of Dibenzo[b,f]oxepines and Total Synthesis of Bauhinoxepin C
40. Tumor‐agnostic inhibitors in oncology: A new phase for precision medicine
41. Synthesis and anti-viral activity of a series of sesquiterpene lactones and analogues in the subgenomic HCV replicon system
42. Overcoming vincristine resistance in cancer: Computational design and discovery of piperine‐inspired P‐glycoprotein inhibitors
43. Drug-like property optimization: Discovery of orally bioavailable quinazoline-based multi-targeted kinase inhibitors
44. A selective Aurora-A 5′-UTR siRNA inhibits tumor growth and metastasis
45. Identification of novel quinoline inhibitor for EHMT2/G9a through virtual screening
46. Lysosomal cysteine protease cathepsin S is involved in cancer cell motility by regulating store-operated Ca2+ entry
47. BPR2-D2 targeting viral ribonucleoprotein complex-associated function inhibits oseltamivir-resistant influenza viruses
48. Bioassay-Guided Purification and Identification of PPARα/γ Agonists from Chlorella sorokiniana
49. Thiopurine analogues inhibit papain-like protease of severe acute respiratory syndrome coronavirus
50. A novel bis-benzylidenecyclopentanone derivative, BPR0Y007, inducing a rapid caspase activation involving upregulation of Fas (CD95/APO-1) and wild-type p53 in human oral epidermoid carcinoma cells
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