2,277 results on '"Hruby, Victor J."'
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2. Melanocortin 3 receptor activation with [D-Trp8]-γ-MSH suppresses inflammation in apolipoprotein E deficient mice
3. Multivalent peptide and peptidomimetic ligands for the treatment of pain without toxicities and addiction
4. Replacement of Arg with Nle and modified D-Phe in the core sequence of MSHs, Ac-His-D-Phe-Arg-Trp-NH2, leads to hMC1R selectivity and pigmentation
5. The Melanocortin-1 Receptor Gene Mediates Female-Specific Mechanisms of Analgesia in Mice and Humans
6. Ψ and χ Angle Constrains at the C-Terminus Trp Position of the Melanotropin Tetrapeptide Ac-His-d-Phe-Arg-Trp-NH2 Lead to Potent and Selective Agonists at hMC1R and hMC4R
7. Melanotropic Peptide-Conjugated Beads for Microscopic Visualization and Characterization of Melanoma Melanotropin Receptors
8. Design synthesis and structure–activity relationship of 5-substituted (tetrahydronaphthalen-2yl)methyl with N-phenyl-N-(piperidin-2-yl)propionamide derivatives as opioid ligands
9. Melanocortin receptors in GtoPdb v.2023.1
10. Supplementary Figures 1-6 from Enhanced targeting with heterobivalent ligands
11. Supplementary Table S1 from Gene expression profiling-based identification of cell-surface targets for developing multimeric ligands in pancreatic cancer
12. Data from Gene expression profiling-based identification of cell-surface targets for developing multimeric ligands in pancreatic cancer
13. Discovery of 5-substituted tetrahydronaphthalen-2yl-methyl with N-phenyl-N-(piperidin-4-yl)propionamide derivatives as potent opioid receptor ligands
14. Design, synthesis, and biological evaluation of a series of bifunctional ligands of opioids/SSRIs
15. Delta Opioid Receptor Function
16. Simple size-selective separation and microscopic characterization of Phe–Phe nanotubes and study of its internalization inside CHO cells
17. Synthesis and evaluation of bivalent ligands for binding to the human melanocortin-4 receptor
18. Melanotropin Receptors and Signal Transduction
19. Cyclic, Conformationally Constrained Melanotropin Analogs: Structure-Function and Conformational Relationships
20. Melanotropin Three-Dimensional Structural Studies by Physical Methods and Computer-Assisted Molecular Modeling
21. New Paradigms and Tools in Drug Design for Pain and Addiction
22. Adjuvants in Cancer Vaccines - Progress and Challenges
23. Examination of the Role of Lipid Rafts in GPCR Signal Transduction Using Plasmon Waveguide Resonance (PWR) Spectroscopy
24. Novel fentanyl-based dual μ/δ-opioid agonists for the treatment of acute and chronic pain
25. Synthesis and Characterization of Time-resolved Fluorescence Probes for Evaluation of Competitive Binding to Melanocortin Receptors
26. Perspectives for the new peptide millennium
27. Design of a δ opioid peptide mimetic based on a topographically constrained cyclic enkephalin
28. Protection against β‐amyloid neurotoxicity by a non‐toxic endogenous N‐terminal β‐amyloid fragment and its active hexapeptide core sequence
29. The Molecular Pharmacology of Alpha-Melanocyte Stimulating Hormone : Structure—Activity Relationships for Melanotropins at Melanocortin Receptors
30. New Perspective in Peptide Chemistry by N-Alkylation
31. Ψ and χ Angle Constrains at the C‑Terminus Trp Position of the Melanotropin Tetrapeptide Ac-His‑d‑Phe-Arg-Trp-NH2 Lead to Potent and Selective Agonists at hMC1R and hMC4R.
32. Heterobivalent ligands target cell-surface receptor combinations in vivo
33. Tachykinin NK1 receptor antagonist co-administration attenuates opioid withdrawal-mediated spinal microglia and astrocyte activation
34. MC4R biased signalling and the conformational basis of biological function selections
35. The Potential Application of Melanotropin Ligands for the Treatment of Obesity and Related Disorders: Potential and Problems
36. Discovery and Development of Novel Melanogenic Drugs : Melanotan-I and -II
37. Design, Synthesis, and Evaluation of Piperazine-Based Small Molecule Peptide Mimetics Targeting the Melanocortin Receptors
38. Understanding BBB Transport using Glycosylated Enkephalins and Endorphins
39. Synthesis and biological evaluation of new opioid agonist and neurokinin-1 antagonist bivalent ligands
40. Conformational study on cyclic melanocortin ligands and new insight into their binding mode at the MC4 receptor
41. Improved synthesis of d, l-fluorocitric acid
42. Utilize conjugated melanotropins for the earlier diagnosis and treatment of melanoma
43. Design of novel melanocortin receptor ligands: Multiple receptors, complex pharmacology, the challenge
44. Novel peptide ligands with dual acting pharmacophores designed for the pathophysiology of neuropathic pain
45. CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists
46. The Design and Synthesis of Long-Acting Oxytocin Antagonists Substituted in Positions 2, 7, and 8
47. Practical glycopeptide analgesics: Blood-brain barrier transport and binding of glycosylated enkephalin analogs
48. Efficacy: What is it, and why you should care
49. Stereoselective synthesis of highly topographically constrained β-isopropyl substituted aromatic amino acids
50. Design of novel melanotropin antagonists and agonists for the recently discovered MC3, MC4 and MC5 receptors and their use to determine new biological roles
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