38 results on '"Gagne, Didier"'
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2. Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor : Gq complex
3. The novel nonapeptide acein targets angiotensin converting enzyme in the brain and induces dopamine release
4. Involvement of tryptophan W276 and of two surrounding amino acid residues in the high constitutive activity of the ghrelin receptor GHS-R1a
5. Regulation of ERK1/2 activity by ghrelin-activated growth hormone secretagogue receptor 1A involves a PLC/PKCε pathway
6. Cholecystokinin 1 receptor modulates the MEKK1-induced c-Jun trans-activation: structural requirements of the receptor
7. New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center
8. Chemical labeling associated to Mass spectrometry as a powerful tool for peptide detection and quantification in biology
9. New trisubstituted 1,2,4-triazoles as ghrelin receptor antagonists
10. Measuring molecular interactions in pharmacological assays by mass spectrometryMeasuring molecular interactions in pharmacological assays by mass spectrometry
11. Quantitative MALDI‐MS Binding Assays: An Alternative to Radiolabeling
12. Selective homodimerization of unprotected peptides using hybrid hydroxydimethylsilane derivatives
13. GHSR-D2R heteromerization modulates dopamine signaling through an effect on G protein conformation.
14. Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
15. Novel Non-Peptide Ghrelin Receptor Ligands Based on 3,4,5-Trisubstituted 1,2,4-triazoles
16. Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex
17. Ghrelin ligands : from design and synthesis to clinical studies
18. Replacement of the alpha-aminoisobutyyl Moiety to obtain Potent Ghrelin Receptor 1,2,4-triazole Based Ligands
19. Cooperation Between GHS-Rla and GHS-Rlb : Action on MAPkinase Pathway
20. New series of Ghrelin Receptor Ligands : Structure Activity Relationship Study on the triazole Moiety
21. Design of Ghrelin Receptor Ligands : From Peptides to Peptidomimetics
22. Synthesis and Biological Evaluations of Ghrelin Ligands
23. Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a
24. Activation of the Ghrelin Receptor is Described by a Privileged Collective Motion: A Model for Constitutive and Agonist-induced Activation of a Sub-class A G-Protein Coupled Receptor (GPCR)
25. C-terminal heptapeptide of gastrin inhibits astrocytomas motility by interacting with a new gastrin binding site.
26. New Trisubstituted 1,2,4-Triazole Derivatives as Potent Ghrelin Receptor Antagonists. 3. Synthesis and Pharmacological in Vitro and in Vivo Evaluations
27. Toward Potent Ghrelin Receptor Ligands Based on Trisubstituted 1,2,4-Triazole Structure. 2. Synthesis and Pharmacological in Vitro and in Vivo Evaluations
28. Synthesis and Pharmacological in Vitro and in Vivo Evaluations of Novel Triazole Derivatives as Ligands of the Ghrelin Receptor. 1
29. Cross-interactions of Two p38 Mitogen-activated Protein (MAP) Kinase Inhibitors and Two Cholecystokinin (CCK) Receptor Antagonists with the CCK1 Receptor and P38 MAP Kinase
30. C-Terminal Heptapeptide of Gastrin Inhibits Astrocytomas Motility by Interacting with a New Gastrin Binding Site
31. The Third Intracellular Loop of the Rat and Mouse Cholecystokinin-A Receptors Is Responsible for Different Patterns of Gene Activation
32. CholecystokininBReceptor from Human Jurkat Lymphoblastic T Cells Is Involved in Activator Protein-1-Responsive Gene Activation
33. Stable luciferase transfected cells for studying steroid receptor biological activity
34. MVLN Cells: A bioluminescent MCF-7-derived cell line to study the modulation of estrogenic activity
35. Study of an antiestrogenic effect of retinoic acid in MCF-7 cells
36. Analysis of the relation between receptor binding affinity and antagonist efficacy of antiglucocorticoids
37. A model of antiglucocorticoid action for designing a potent glucocorticoid antagonist
38. Description and analysis of differential sensitivity to glucocorticoids in Fao cells
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