48 results on '"Centrella, Paolo A."'
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2. Novel irreversible covalent BTK inhibitors discovered using DNA-encoded chemistry
3. Discovery of soluble epoxide hydrolase inhibitors through DNA-encoded library technology (ELT)
4. Rational Design of Macrocyclic Noncovalent Inhibitors of SARS-CoV-2 Mprofrom a DNA-Encoded Chemical Library Screening Hit That Demonstrate Potent Inhibition against Pan-Coronavirus Homologues and Nirmatrelvir-Resistant Variants
5. A resource to enable chemical biology and drug discovery of WDR Proteins
6. Development of Potent Mcl-1 Inhibitors: Structural Investigations on Macrocycles Originating from a DNA-Encoded Chemical Library Screen
7. Discovery of a First-in-Class Small-Molecule Ligand for WDR91 Using DNA-Encoded Chemical Library Selection Followed by Machine Learning
8. Agonists and Antagonists of Protease-Activated Receptor 2 Discovered within a DNA-Encoded Chemical Library Using Mutational Stabilization of the Target
9. Discovery of cofactor-specific, bactericidal Mycobacterium tuberculosis InhA inhibitors using DNA-encoded library technology
10. Discovery of Small Molecule Interleukin 17A Inhibitors with Novel Binding Mode and Stoichiometry: Optimization of DNA-Encoded Chemical Library Hits to In Vivo Active Compounds
11. Abstract 5331: DNA-encoded macrocyclic compound libraries for challenging targets
12. Correction: Author Correction: Prioritizing multiple therapeutic targets in parallel using automated DNA-encoded library screening
13. Discovery of Novel UDP-N-Acetylglucosamine Acyltransferase (LpxA) Inhibitors with Activity against Pseudomonas aeruginosa
14. Design, synthesis and selection of DNA-encoded small-molecule libraries
15. Discovery of Novel, Potent Inhibitors of Hydroxy Acid Oxidase 1 (HAO1) Using DNA-Encoded Chemical Library Screening
16. Novel Nucleic Acid Binding Small Molecules Discovered Using DNA-Encoded Chemistry
17. Development and Synthesis of DNA-Encoded Benzimidazole Library
18. Corrigendum: Discovery of a Potent BTK Inhibitor with a Novel Binding Mode by Using Parallel Selections with a DNAEncoded Chemical Library
19. Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action
20. Correction to “Structure Based Design of Non-Natural Peptidic Macrocyclic Mcl-1 Inhibitors”
21. Prioritizing multiple therapeutic targets in parallel using automated DNA-encoded library screening
22. Abstract 5084: Potent and isoform-selective ATAD2 bromodomain inhibitor with unprecedented chemical structure and mode of action
23. Inside Cover: Discovery of a Potent BTK Inhibitor with a Novel Binding Mode by Using Parallel Selections with a DNA-Encoded Chemical Library (ChemBioChem 9/2017)
24. Discovery of a Potent BTK Inhibitor with a Novel Binding Mode by Using Parallel Selections with a DNA-Encoded Chemical Library
25. Structure Based Design of Non-Natural Peptidic Macrocyclic Mcl-1 Inhibitors
26. Design and Synthesis of Biaryl DNA-Encoded Libraries
27. Development and Synthesis of DNA-Encoded Benzimidazole Library.
28. A Target Class Ligandability Evaluation of WD40 Repeat-Containing Proteins
29. Cell-Based Selection Expands the Utility of DNA-Encoded Small-Molecule Library Technology to Cell Surface Drug Targets: Identification of Novel Antagonists of the NK3 Tachykinin Receptor
30. Discovery, SAR, and X-ray Binding Mode Study of BCATm Inhibitors from a Novel DNA-Encoded Library
31. Encoded Library Synthesis Using Chemical Ligation and the Discovery of sEH Inhibitors from a 334-Million Member Library
32. Discovery of a Potent Class of PI3Kα Inhibitors with Unique Binding Mode via Encoded Library Technology (ELT)
33. Encoded Library Technology as a Source of Hits for the Discovery and Lead Optimization of a Potent and Selective Class of Bactericidal Direct Inhibitors of Mycobacterium tuberculosis InhA
34. Antiparasitic activities of novel, orally available fumagillin analogs
35. Orally Active Fumagillin Analogues: Transformations of a Reactive Warhead in the Gastric Environment
36. Design and Synthesis of Biaryl DNA-Encoded Libraries.
37. Metabolites of PPI-2458, a Selective, Irreversible Inhibitor of Methionine Aminopeptidase-2: Structure Determination and In Vivo Activity
38. Discovery of Highly Potent and Selective Small Molecule ADAMTS-5 Inhibitors That Inhibit Human Cartilage Degradation via Encoded Library Technology (ELT)
39. Carbamate Analogues of Fumagillin as Potent, Targeted Inhibitors of Methionine Aminopeptidase-2
40. Erratum: Design, synthesis and selection of DNA-encoded small-molecule libraries
41. Cell-Based Selection Expands the Utility of DNA-Encoded Small-Molecule Library Technology to Cell Surface Drug Targets: Identification of Novel Antagonists of the NK3 Tachykinin Receptor.
42. Encoded Library Technologyas a Source of Hits forthe Discovery and Lead Optimization of a Potent and Selective Classof Bactericidal Direct Inhibitors of Mycobacterium tuberculosisInhA.
43. Discovery of Highly Potentand Selective Small MoleculeADAMTS-5 Inhibitors That Inhibit Human Cartilage Degradationvia Encoded Library Technology (ELT).
44. Author Correction: Prioritizing multiple therapeutic targets in parallel using automated DNA-encoded library screening.
45. Rational Design of Macrocyclic Noncovalent Inhibitors of SARS-CoV-2 M pro from a DNA-Encoded Chemical Library Screening Hit That Demonstrate Potent Inhibition against Pan-Coronavirus Homologues and Nirmatrelvir-Resistant Variants.
46. Identification and Evaluation of Reversible Covalent Binders to Cys55 of Bfl-1 from a DNA-Encoded Chemical Library Screen.
47. Inhibitors of the Thioesterase Activity of Mycobacterium tuberculosis Pks13 Discovered Using DNA-Encoded Chemical Library Screening.
48. Structure Based Design of Non-Natural Peptidic Macrocyclic Mcl-1 Inhibitors.
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