198 results on '"Brussee, Johannes"'
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2. Dual-Point Competition Association Assay: A Fast and High-Throughput Kinetic Screening Method for Assessing Ligand-Receptor Binding Kinetics
3. Stereoselective Biocatalytic Formation of Cyanohydrins, Versatile Building Blocks for Organic Synthesis
4. Synthesis and biological evaluation of 2-aminothiazoles and their amide derivatives on human adenosine receptors. Lack of effect of 2-aminothiazoles as allosteric enhancers
5. Biocatalysis in the Enantioselective Formation of Chiral Cyanohydrins, Valuable Building Blocks in Organic Synthesis
6. Stereoselective Biocatalytic Formation of Cyanohydrins, Versatile Building Blocks for Organic Synthesis
7. Synthesis and biological evaluation of disubstituted N6-cyclopentyladenine analogues: the search for a neutral antagonist with high affinity for the adenosine A1 receptor
8. Conversion of chiral unsaturated cyanohydrins into chiral carba- and heterocycles via ring-closing metathesis
9. Intramolecular reductive cleavage of tert-butyldimethylsilyl ethers. Selective mono-deprotection of bis-silyl-protected diols
10. Synthesis of chiral diaza-18-crown-6 derivatives from optically active diethanolamines
11. Synthesis of Fmoc-protected (2 S,3 S)-2-hydroxy-3-amino acids from a furyl substituted chiral cyanohydrin
12. Mass transfer limitation as a tool to enhance the enantiomeric excess in the enzymatic synthesis of chiral cyanohydrins
13. Synthesis of γ-Hydroxy-α,β-unsaturated Esters and Nitriles from Chiral Cyanohydrins
14. Diastereoselective addition of HCN to Garner's aldehyde
15. Synthesis of reduced collagen crosslinks
16. Evaluation of (4‐Arylpiperidin‐1‐yl)cyclopentanecarboxamides As High‐Affinity and Long‐Residence‐Time Antagonists for the CCR2 Receptor
17. Agonists for the Adenosine A1 Receptor with Tunable Residence Time. A Case for Nonribose 4-Amino-6-aryl-5-cyano-2-thiopyrimidines
18. Binding Kinetics of ZM241385 Derivatives at the Human Adenosine A2AReceptor
19. Synthesis of Eight 1-Deoxynojirimycin Isomers from a Single Chiral Cyanohydrin
20. Removal of Human Ether-à-go-go Related Gene (hERG) K+ Channel Affinity through Rigidity: A Case of Clofilium Analogues
21. Structure–Kinetic Relationships—An Overlooked Parameter in Hit-to-Lead Optimization: A Case of Cyclopentylamines as Chemokine Receptor 2 Antagonists
22. Strategies To Reduce hERG K+Channel Blockade. Exploring Heteroaromaticity and Rigidity in Novel Pyridine Analogues of Dofetilide
23. Multi-Objective Evolutionary Design of Adenosine Receptor Ligands
24. Synthesis of Eight 1-Deoxynojirimycin Isomers from a Single Chiral Cyanohydrin
25. Determination of different putative allosteric binding pockets at the lutropin receptor by using diverse drug-like low molecular weight ligands
26. Novel 3,6,7-Substituted Pyrazolopyrimidines as Positive Allosteric Modulators for the Hydroxycarboxylic Acid Receptor 2 (GPR109A)
27. Cover Picture: Understanding of Molecular Substructures that Contribute to hERG K+ Channel Blockade: Synthesis and Biological Evaluation of E‐4031 Analogues (ChemMedChem 1/2012)
28. Understanding of Molecular Substructures that Contribute to hERG K+ Channel Blockade: Synthesis and Biological Evaluation of E‐4031 Analogues
29. Synthesis of l-altro-1-Deoxynojirimycin, d-allo-1-Deoxynojirimycin, and d-galacto-1-Deoxynojirimycin from a Single Chiral Cyanohydrin
30. ChemInform Abstract: Synthesis of Reduced Collagen Crosslinks.
31. ChemInform Abstract: Synthesis of γ-Hydroxy-α,β-unsaturated Esters and Nitriles from Chiral Cyanohydrins.
32. ChemInform Abstract: Biocatalysis in the Enantioselective Formation of Chiral Cyanohydrins, Valuable Building Blocks in Organic Synthesis
33. ChemInform Abstract: Stereoselective Biocatalytic Formation of Cyanohydrins, Versatile Building Blocks for Organic Synthesis
34. Hybrid Ortho/Allosteric Ligands for the Adenosine A1 Receptor
35. Corrections to Substituted Terphenyl Compounds as the First Class of Low Molecular Weight Allosteric Inhibitors of the Luteinizing Hormone Receptor
36. Substituted Terphenyl Compounds as the First Class of Low Molecular Weight Allosteric Inhibitors of the Luteinizing Hormone Receptor
37. A Series of 2,4-Disubstituted Quinolines as a New Class of Allosteric Enhancers of the Adenosine A3 Receptor
38. False Positives in a Reporter Gene Assay: Identification and Synthesis of Substituted N-Pyridin-2-ylbenzamides as Competitive Inhibitors of Firefly Luciferase
39. 2-Amino-6-furan-2-yl-4-substituted Nicotinonitriles as A2A Adenosine Receptor Antagonists
40. A new generation of adenosine receptor antagonists: From di- to trisubstituted aminopyrimidines
41. Designing Active Template Molecules by Combining Computational De Novo Design and Human Chemist's Expertise
42. 2,6,8-Trisubstituted 1-Deazapurines as Adenosine Receptor Antagonists
43. Structure−Activity Relationships of New 1H-Imidazo[4,5-c]quinolin-4-amine Derivatives as Allosteric Enhancers of the A3 Adenosine Receptor
44. 2,6-Disubstituted and 2,6,8-Trisubstituted Purines as Adenosine Receptor Antagonists
45. Conversion of Chiral Unsaturated Cyanohydrins into Chiral Carba- and Heterocycles via Ring-Closing Metathesis.
46. Synthesis and Biological Evaluation of a New Series of 2,3,5-Substituted [1,2,4]-Thiadiazoles as Modulators of Adenosine A1 Receptors and Their Molecular Mechanism of Action
47. 2,4,6-Trisubstituted Pyrimidines as a New Class of Selective Adenosine A1 Receptor Antagonists
48. Non-Xanthine Antagonists for the Adenosine A1 Receptor
49. A Series of Ligands Displaying a Remarkable Agonistic−Antagonistic Profile at the Adenosine A1 Receptor
50. New, Non-Adenosine, High-Potency Agonists for the Human Adenosine A2B Receptor with an Improved Selectivity Profile Compared to the Reference Agonist N-Ethylcarboxamidoadenosine
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