268 results on '"Bathgate, Ross A.D."'
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2. Modulation of contextual fear acquisition and extinction by acute and chronic relaxin-3 receptor (RXFP3) activation in the rat retrosplenial cortex
3. Developing insulin-like peptide 5-based antagonists for the G protein-coupled receptor, RXFP4
4. Development of a synthetic relaxin-3/INSL5 chimeric peptide ligand for NanoBiT complementation binding assays
5. The single-chain relaxin mimetic, B7-33, maintains the cardioprotective effects of relaxin and more rapidly reduces left ventricular fibrosis compared to perindopril in an experimental model of cardiomyopathy
6. Ligands selectively tune the local and global motions of neurotensin receptor 1 (NTS1)
7. Spawning induction of the high-value white teatfish sea cucumber, Holothuria fuscogilva, using recombinant relaxin-like gonad stimulating peptide (RGP)
8. Structural Insights into the Unique Modes of Relaxin-Binding and Tethered-Agonist Mediated Activation of RXFP1 and RXFP2
9. Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists
10. A Chemogenetic Tool that Enables Functional Neural Circuit Analysis
11. Targeted viral vector transduction of relaxin-3 neurons in the rat nucleus incertus using a novel cell-type specific promoter
12. Probing the correlation between ligand efficacy and conformational diversity at the α1A-adrenoreceptor reveals allosteric coupling of its microswitches
13. An apically located hybrid guanylate cyclase–ATPase is critical for the initiation of Ca2+ signaling and motility in Toxoplasma gondii
14. Identification of a Novel Subtype-Selective α1B-Adrenoceptor Antagonist
15. Multi-Component Mechanism of H2 Relaxin Binding to RXFP1 through NanoBRET Kinetic Analysis
16. Distinct but overlapping binding sites of agonist and antagonist at the relaxin family peptide 3 (RXFP3) receptor
17. Binding conformation and determinants of a single-chain peptide antagonist at the relaxin-3 receptor RXFP3
18. The relaxin receptor as a therapeutic target – perspectives from evolution and drug targeting
19. Challenges in the design of insulin and relaxin/insulin-like peptide mimetics
20. Optimization and 13CH3 methionine labeling of a signaling competent neurotensin receptor 1 variant for NMR studies
21. B7-33 replicates the vasoprotective functions of human relaxin-2 (serelaxin)
22. Bi-allelic variants in INSL3 and RXFP2 cause bilateral cryptorchidism and male infertility
23. Identification of a Novel Subtype-Selective α1B-Adrenoceptor Antagonist.
24. Relaxin family peptide receptors in GtoPdb v.2023.1
25. Investigation of Interactions at the Extracellular Loops of the Relaxin Family Peptide Receptor 1 (RXFP1)
26. Improving the apo-state detergent stability of NTS1 with CHESS for pharmacological and structural studies
27. Relaxin requires the angiotensin II type 2 receptor to abrogate renal interstitial fibrosis
28. The Relaxin Receptor (RXFP1) Utilizes Hydrophobic Moieties on a Signaling Surface of Its N-terminal Low Density Lipoprotein Class A Module to Mediate Receptor Activation
29. Identification of Key Residues Essential for the Structural Fold and Receptor Selectivity within the A-chain of Human Gene-2 (H2) Relaxin
30. Chimeric relaxin peptides highlight the role of the A-chain in the function of H2 relaxin
31. A unique peptide recognition mechanism by the human relaxin family peptide receptor 4 (RXFP4)
32. The Minimal Active Structure of Human Relaxin-2
33. Membrane receptors: Structure and function of the relaxin family peptide receptors
34. A simple approach for the preparation of mature human relaxin-3
35. Role of the intra-A-chain disulfide bond of insulin-like peptide 3 in binding and activation of its receptor, RXFP2
36. Swim stress excitation of nucleus incertus and rapid induction of relaxin-3 expression via CRF 1 activation
37. High-Throughput Screening Campaign Identified a Potential Small Molecule RXFP3/4 Agonist
38. Ligand recognition mechanism of the human relaxin family peptide receptor 4 (RXFP4)
39. Structure of the R3/I5 Chimeric Relaxin Peptide, a Selective GPCR135 and GPCR142 Agonist
40. The A-chain of Human Relaxin Family Peptides Has Distinct Roles in the Binding and Activation of the Different Relaxin Family Peptide Receptors
41. Relaxin family peptide receptors – from orphans to therapeutic targets
42. Negative cooperativity in H2 relaxin binding to a dimeric relaxin family peptide receptor 1
43. Prolonged RXFP1 and RXFP2 signaling can be explained by poor internalization and a lack of [beta]-arrestin recruitment
44. R3(BΔ23–27)R/I5 Chimeric Peptide, a Selective Antagonist for GPCR135 and GPCR142 over Relaxin Receptor LGR7: IN VITRO AND IN VIVO CHARACTERIZATION
45. Improved chemical synthesis and demonstration of the relaxin receptor binding affinity and biological activity of mouse relaxin
46. The NMR Solution Structure of the Relaxin (RXFP1) Receptor Lipoprotein Receptor Class A Module and Identification of Key Residues in the N-terminal Region of the Module That Mediate Receptor Activation
47. Comparison of Signaling Pathways Activated by the Relaxin Family Peptide Receptors, RXFP1 and RXFP2, Using Reporter Genes
48. Paracrine regulation of mammalian oocyte maturation and male germ cell survival
49. Characterization of Novel Splice Variants of LGR7 and LGR8 Reveals That Receptor Signaling Is Mediated by Their Unique Low Density Lipoprotein Class A Modules
50. Solution Structure and Characterization of the LGR8 Receptor Binding Surface of Insulin-like Peptide 3
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