469 results on '"Arora, Paramjit"'
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2. A Sos proteomimetic as a pan-Ras inhibitor
3. Targeting the succinate receptor effectively inhibits periodontitis
4. C2230, A Selective, Use- And State-Dependent CaV2.2 Channel Blocker for Neuropathic, Orofacial, and Osteoarthritic Pain
5. Hydrogen bond surrogate helices as minimal mimics of protein α-helices
6. Hydrogen Bond Surrogate Stabilized Helices as Protein–Protein Interaction Inhibitors
7. An Encodable Scaffold for Sequence‐Specific Recognition of Duplex RNA
8. Oligooxopiperazines as Topographical Helix Mimetics
9. Macrocyclic β‐Sheets Stabilized by Hydrogen Bond Surrogates
10. Comparative ACE2 variation and primate COVID-19 risk
11. Modulation of virus-induced NF-κB signaling by NEMO coiled coil mimics
12. A Selective Peptidomimetic Modulator Of Cav2.2 (N-Type) Voltage-Gated Calcium Channels For Chronic Pain
13. Structure-based inhibition of protein–protein interactions
14. Rational Design Strategies for Developing Synthetic Inhibitors of Helical Protein Interfaces
15. Late‐Stage Modification of Oligopeptides by Nickel‐Catalyzed Stereoselective Radical Addition to Dehydroalanine
16. Anchor Residues Govern Binding and Folding of an Intrinsically Disordered Domain
17. A rationally designed peptidomimetic modulator of CaV2.2 (N-type) voltage-gated calcium channels for chronic pain
18. Variation in predicted COVID-19 risk among lemurs and lorises
19. In vivo modulation of hypoxia-inducible signaling by topographical helix mimetics
20. Effects of side chains in helix nucleation differ from helix propagation
21. Modeling and Design of Peptidomimetics to Modulate Protein–Protein Interactions
22. Variation in predicted COVID-19 risk among lemurs and lorises
23. Plucking the high hanging fruit: A systematic approach for targeting protein–protein interactions
24. Protein domain mimetics as in vivo modulators of hypoxia-inducible factor signaling
25. Reversible α-helix formation controlled by a hydrogen bond surrogate
26. End-capped α-helices as modulators of protein function
27. Oligooxopiperazines as Topographical Helix Mimetics
28. Peptide Tethering: Pocket-Directed Fragment Screening for Peptidomimetic Inhibitor Discovery
29. Design and Synthesis of Crosslinked Helix Dimers as Protein Tertiary Structure Mimics
30. Targeting Succinate Receptor Reduces Microglial Activation and Neuroinflammation
31. Covalent and Noncovalent Targeting of the Tcf4/β-Catenin Strand Interface with β-Hairpin Mimics
32. Identification of Secondary Binding Sites on Protein Surfaces for Rational Elaboration of Synthetic Protein Mimics
33. Dual Control of Peptide Conformation with Light and Metal Coordination
34. Contemporary strategies for the stabilization of peptides in the α-helical conformation
35. Variation in predicted COVID‐19 risk among lemurs and lorises
36. HippDB: a database of readily targeted helical protein–protein interactions
37. An Orthosteric Inhibitor of the RAS–SOS Interaction
38. Conformational control in a photoswitchable coiled coil
39. Daniel S. Kemp (1936–2020): A Pioneer of Bioorganic Chemistry
40. Faculty Opinions recommendation of Phosphorylation-Inducing Chimeric Small Molecules.
41. Faculty Opinions recommendation of Design, synthesis and characterization of structurally dynamic cyclic N,S-acetals.
42. Macropinocytosis as a Key Determinant of Peptidomimetic Uptake in Cancer Cells
43. Faculty Opinions recommendation of Efficient targeted degradation via reversible and irreversible covalent protacs.
44. Faculty Opinions recommendation of An azidoribose probe to track ketoamine adducts in histone ribose glycation.
45. Faculty Opinions recommendation of Small-molecule covalent bond formation at tyrosine creates a binding site and inhibits activation of Ral GTPases.
46. Covalent Targeting of Ras G12C by Rationally Designed Peptidomimetics
47. Comparative ACE2 variation and primate COVID-19 risk
48. Bent into shape: Folded peptides to mimic protein structure and modulate protein function
49. Faculty Opinions recommendation of The Bioorthogonal Isonitrile-Chlorooxime Ligation.
50. Faculty Opinions recommendation of Global targeting of functional tyrosines using sulfur-triazole exchange chemistry.
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