286 results on '"Addlagatta, Anthony"'
Search Results
2. Anti-inflammatory and antioxidant activities of Gymnema Sylvestre extract rescue acute respiratory distress syndrome in rats via modulating the NF-κB/MAPK pathway
3. A single amino acid difference between archaeal and human type 2 methionine aminopeptidases differentiates their affinity towards ovalicin
4. Regioselectivity in inhibition of peptide deformylase from Haemophilus influenzae by 4- vs 5-azaindole hydroxamic acid derivatives: Biochemical, structural and antimicrobial studies
5. Benzothiazolo-quinazoline Congeners Function as Anti-microtubule Agents Triggering Mitotic Arrest in Cancer Cells
6. Selective inhibition of Helicobacter pylori methionine aminopeptidase by azaindole hydroxamic acid derivatives: Design, synthesis, in vitro biochemical and structural studies
7. Methionine aminopeptidases with short sequence inserts within the catalytic domain are differentially inhibited: Structural and biochemical studies of three proteins from Vibrio spp.
8. Strategic enzymatic enantioselective desymmetrization of prochiral cyclohexa-2,5-dienones.
9. Exo-selective intermolecular Diels–Alder reaction by PyrI4 and AbnU on non-natural substrates
10. Synthesis and mechanistic studies of diketo acids and their bioisosteres as potential antibacterial agents
11. Gymnema sylvestre extract improves PCOS by altering the YAP1 protein in the mouse ovary via mitochondrial changes
12. Development of 2-chloroquinoline based heterocyclic frameworks as dual inhibitors of SARS-CoV-2 MPro and PLPro
13. Inhibition of Xanthine oxidase by 1-O-methyl chrysophanol, a hydroxyanthraquinone isolated fromAmycolatopsis thermoflavaICTA 103
14. Highly functionalized tetrahydropyridines are cytotoxic and selective inhibitors of human puromycin sensitive aminopeptidase
15. Bengamides display potent activity against drug-resistant Mycobacterium tuberculosis
16. Design and synthesis of pyrazole–oxindole conjugates targeting tubulin polymerization as new anticancer agents
17. Synthesis and structure–activity relationships of pyridinyl-1H-1,2,3-triazolyldihydroisoxazoles as potent inhibitors of tubulin polymerization
18. Discovery of Tröger's base analogues as selective inhibitors against human breast cancer cell line: Design, synthesis and cytotoxic evaluation
19. Expression, Functional Characterization and X-ray Analysis of HosA, A Member of MarR Family of Transcription Regulator from Uropathogenic Escherichia coli
20. Design, Synthesis and Mechanistic Studies of Novel Isatin-Pyrazole Hydrazone Conjugates as Selective and Potent Bacterial MetAP Inhibitors
21. Anti-inflammatory and anti-oxidant activities of Gymnema sylvestre extract rescues acute respiratory distress syndrome in rats via modulating the NF-κB/MAPK pathway
22. Design and synthesis of biaryl aryl stilbenes/ethylenes as antimicrotubule agents
23. Design, Synthesis and Mechanistic Studies of Novel Isatin-Pyrazole Hydrazone Conjugates as Selective and Potent Bacterial MetAP Inhibitors
24. Genomic characterization and evolutionary analysis of dengue virus from Aedes mosquitoes in Telangana, India.
25. Synthesis and biological evaluation of combretastatin-amidobenzothiazole conjugates as potential anticancer agents
26. Synthesis of chalcone-amidobenzothiazole conjugates as antimitotic and apoptotic inducing agents
27. Development of peptidomimetic hydroxamates as PfA-M1 and PfA-M17 dual inhibitors: Biological evaluation and structural characterization by cocrystallization
28. Genomic characterization and evolutionary analysis of dengue virus from Aedes mosquitoes in Telangana, India
29. Elucidation of the Function of Type 1 Human Methionine Aminopeptidase during Cell Cycle Progression
30. Structure of Aminopeptidase N from Escherichia coli Suggests a Compartmentalized, Gated Active Site
31. Pancreatic α-amylase inhibition and free radical scavenging activity of substituted pyranochromenone derivatives
32. Structure activity relationship studies of imidazo[1,2-a]pyrazine derivatives against cancer cell lines
33. Chemical shift assignments of zinc finger domain of methionine aminopeptidase 1 (MetAP1) from Homo sapiens
34. Structural basis for the inhibition of M1 family aminopeptidases by the natural product actinonin: Crystal structure in complex with E. coli aminopeptidase N
35. Structural characterization of the protein cce_0567 from Cyanothece 51142, a metalloprotein associated with nitrogen fixation in the DUF683 family
36. Selective targeting of the conserved active site cysteine of Mycobacterium tuberculosis methionine aminopeptidase with electrophilic reagents
37. Structural basis for the functional difference between type I and type II human methionine aminopeptidases
38. Puromycin, a selective inhibitor of PSA acts as a substrate for other M1 family aminopeptidases: Biochemical and structural basis
39. Glu121-Lys319 salt bridge between catalytic and N-terminal domains is pivotal for the activity and stability of Escherichia coli aminopeptidase N
40. Structure of the angiogenesis inhibitor ovalicin bound to its noncognate target, human Type 1 methionine aminopeptidase
41. Determining Structure and Function of Steroid Dehydrogenase Enzymes by Sequence Analysis, Homology Modeling, and Rational Mutational Analysis
42. Aminobenzosuberone Scaffold as a Modular Chemical Tool for the Inhibition of Therapeutically Relevant M1 Aminopeptidases
43. Unraveling structural insights of ribokinase from Leishmania donovani
44. Discovery of a new class of type 1 methionine aminopeptidases that have relaxed substrate specificity
45. Discovery of natural product ovalicin sensitive type 1 methionine aminopeptidases: molecular and structural basis
46. Discovery, Structural and Biochemical Studies of a rare Glu/Asp Specific M1 Class Aminopeptidase from Legionella pneumophila
47. Crystal structure and vibrational spectrum of N-methylpiperidine betaine hexafluorosilicate
48. Understanding the structural basis of Legionella pneumophila aminopeptidase N
49. Discovery of new genetic variants of methionine aminopeptidases
50. Development of selective inhibitors against malarial M1 family aminopeptidase
Catalog
Books, media, physical & digital resources
Discovery Service for Jio Institute Digital Library
For full access to our library's resources, please sign in.