276 results on '"Yasgar, Adam"'
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52. Quantitative high-throughput screening identifies cytoprotective molecules that enhance SUMO conjugation via the inhibition of SUMO-specific protease (SENP)2
53. The Tox21 10K Compound Library: Collaborative Chemistry Advancing Toxicology.
54. Canvass: A Crowd-Sourced, Natural Product Screening Library for Exploring Biological Space
55. Testing for drug-human serum albumin binding using fluorescent probes and other methods
56. Discovery of Orally Bioavailable, Quinoline-Based Aldehyde Dehydrogenase 1A1 (ALDH1A1) Inhibitors with Potent Cellular Activity
57. Correction: A High-Content Assay Enables the Automated Screening and Identification of Small Molecules with Specific ALDH1A1-Inhibitory Activity
58. Discovery and optimization of piperazine-1-thiourea-based human phosphoglycerate dehydrogenase inhibitors
59. Quantitative high‐throughput screening identifies cytoprotective molecules that enhance SUMO conjugation via the inhibition of SUMO‐specific protease (SENP)2
60. Parallel Chemistry Approach to Identify Novel Nuclear Receptor Ligands Based on the GW0742 Scaffold
61. Structure–activity relationship studies and biological characterization of human NAD+-dependent 15-hydroxyprostaglandin dehydrogenase inhibitors
62. A High-Content Assay Enables the Automated Screening and Identification of Small Molecules with Specific ALDH1A1-Inhibitory Activity
63. A High-Throughput Screen Identifies 2,9-Diazaspiro[5.5]Undecanes as Inducers of the Endoplasmic Reticulum Stress Response with Cytotoxic Activity in 3D Glioma Cell Models
64. A High-Throughput Screen Identifies 2,9-Diazaspiro[5.5]Undecanes as Inducers of the Endoplasmic Reticulum Stress Response with Cytotoxic Activity in 3D Glioma Cell Models
65. Erratum: Corrigendum: A PHGDH inhibitor reveals coordination of serine synthesis and one-carbon unit fate
66. Fluorescence polarization assays in high-throughput screening and drug discovery: a review
67. A PHGDH inhibitor reveals coordination of serine synthesis and one-carbon unit fate
68. Discovery of Orally Bioavailable, Quinoline-Based Aldehyde Dehydrogenase 1A1 (ALDH1A1) Inhibitors with Potent Cellular Activity.
69. Optimization of High-Throughput Methyltransferase Assays for the Discovery of Small Molecule Inhibitors
70. Discovery of NCT-501, a Potent and Selective Theophylline-Based Inhibitor of Aldehyde Dehydrogenase 1A1 (ALDH1A1)
71. Current approaches for the discovery of drugs that deter substance and drug abuse
72. This title is unavailable for guests, please login to see more information.
73. High-throughput combinatorial screening identifies drugs that cooperate with ibrutinib to kill activated B-cell–like diffuse large B-cell lymphoma cells
74. 4-(3-Chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide (ML267), a Potent Inhibitor of Bacterial Phosphopantetheinyl Transferase That Attenuates Secondary Metabolism and Thwarts Bacterial Growth
75. Synthesis and Structure–Activity Relationship Studies of 4-((2-Hydroxy-3-methoxybenzyl)amino)benzenesulfonamide Derivatives as Potent and Selective Inhibitors of 12-Lipoxygenase
76. Abstract 4543: High-throughput combination screening identifies novel drug-drug pairings for a Bruton's tyrosine kinase inhibitor against the ABC subtype of diffuse large B-cell lymphomas.
77. High-Throughput 1,536-Well Fluorescence Polarization Assays for α1-Acid Glycoprotein and Human Serum Albumin Binding
78. The NCGC Pharmaceutical Collection: A Comprehensive Resource of Clinically Approved Drugs Enabling Repurposing and Chemical Genomics
79. A High-Throughput 1,536-Well Luminescence Assay for Glutathione S-Transferase Activity
80. A strategy to discover inhibitors of Bacillus subtilis surfactin-type phosphopantetheinyl transferase
81. Preparation of FRET reporters to support chemical probe development
82. A High Throughput Fluorescence Polarization Assay for Inhibitors of the GoLoco Motif/G-alpha Interaction
83. Compound Management for Quantitative High-Throughput Screening
84. Evaluation of Micro-Parallel Liquid Chromatography as a Method for HTS-Coupled Actives Verification
85. THE IMPACT OF P-GLYCOPROTEIN ON THE DISPOSITION OF DRUGS TARGETED FOR INDICATIONS OF THE CENTRAL NERVOUS SYSTEM: EVALUATION USING THE MDR1A/1B KNOCKOUT MOUSE MODEL
86. [29] - Fluorescent Protein‐Based Cellular Assays Analyzed by Laser‐Scanning Microplate Cytometry in 1536‐Well Plate Format
87. Biochemical and Cellular Characterization and Inhibitor Discovery of Pseudomonas aeruginosa15-Lipoxygenase
88. Potent and Selective Inhibitorsof Human Reticulocyte12/15-Lipoxygenase as Anti-Stroke Therapies.
89. 4-(3-Chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide(ML267), a Potent Inhibitor of Bacterial Phosphopantetheinyl TransferaseThat Attenuates Secondary Metabolism and Thwarts Bacterial Growth.
90. Synthesis and Structure–ActivityRelationshipStudies of 4-((2-Hydroxy-3-methoxybenzyl)amino)benzenesulfonamideDerivatives as Potent and Selective Inhibitors of 12-Lipoxygenase.
91. High-Throughput 1,536-Well Fluorescence Polarization Assays for α1-Acid Glycoprotein and Human Serum Albumin Binding.
92. The NCGC Pharmaceutical Collection: A Comprehensive Resource of Clinically Approved Drugs Enabling Repurposing and Chemical Genomics.
93. A PHGDH inhibitor reveals coordination of serine synthesis and 1-carbon unit fate
94. The impact of P-glycoprotein on the disposition of drugs targeted for indications of the central nervous system: evaluation using the MDR1A/1B knockout mouse model.
95. Correction: A High-Throughput Screen Identifies 2,9-Diazaspiro[5.5]Undecanes as Inducers of the Endoplasmic Reticulum Stress Response with Cytotoxic Activity in 3D Glioma Cell Models.
96. Corrigendum: A PHGDH inhibitor reveals coordination of serine synthesis and one-carbon unit fate
97. Small-Molecule Disruptors of the Interaction between Calcium- and Integrin-Binding Protein 1 and Integrin α IIb β 3 as Novel Antiplatelet Agents.
98. RALDH1 Inhibition Shows Immunotherapeutic Efficacy in Hepatocellular Carcinoma.
99. Discovery and Optimization of 2 H -1λ 2 -Pyridin-2-one Inhibitors of Mutant Isocitrate Dehydrogenase 1 for the Treatment of Cancer.
100. Applications of Differential Scanning Fluorometry and Related Technologies in Characterization of Protein-Ligand Interactions.
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