507 results on '"Shen, Jingkang"'
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52. Tranylcypromine and 6-trifluoroethyl thienopyrimidine hybrid as LSD1 inhibitor
53. Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases
54. Correction to “Discovery and Optimization of 4,5-Diarylisoxazoles as Potent Dual Inhibitors of Pyruvate Dehydrogenase Kinase and Heat Shock Protein 90”
55. DrugViz: a Cytoscape plugin for visualizing and analyzing small molecule drugs in biological networks
56. Convenient preparation of pinometostat and related 5′-deoxy-5′-amino adenosine derivatives as well as their activity against DOT1L
57. Preparation of 5′-deoxy-5′-amino-5′-C-methyl adenosine derivatives and their activity against DOT1L
58. The Structure of MT189-Tubulin Complex Provides Insights into Drug Design
59. Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors
60. Design and Synthesis of Potent, Selective Inhibitors of Protein Arginine Methyltransferase 4 against Acute Myeloid Leukemia
61. Stereoselective N-glycosylation with N4-acyl cytosines and efficient synthesis of gemcitabine
62. Discovery of a series of dimethoxybenzene FGFR inhibitors with 5H-pyrrolo[2,3-b]pyrazine scaffold: structure–activity relationship, crystal structural characterization and in vivo study
63. BSSF: a fingerprint based ultrafast binding site similarity search and function analysis server
64. Design and synthesis of benzylpiperidine inhibitors targeting the menin–MLL1 interface
65. Formation of 1,3-diazocine by palladium catalyzed C–H arylation
66. Discovery of novel 2-phenyl-imidazo[1,2-a]pyridine analogues targeting tubulin polymerization as antiproliferative agents
67. Design and discovery of new pyrimidine coupled nitrogen aromatic rings as chelating groups of JMJD3 inhibitors
68. Molecular Modeling Studies on Carbazole Carboxamide Based BTK Inhibitors Using Docking and Structure-Based 3D-QSAR
69. Preclinical Evaluation of SCC244 (Glumetinib), a Novel, Potent, and Highly Selective Inhibitor of c-Met in MET-dependent Cancer Models
70. Structure-Based Discovery of a Series of 5H-Pyrrolo[2,3-b]pyrazine FGFR Kinase Inhibitors
71. Efficient syntheses of alpha- and beta-C-nucleosides and the origin of anomeric selectivity
72. Pathological expression of tissue factor confers promising antitumor response to a novel therapeutic antibody SC1 in triple negative breast cancer and pancreatic adenocarcinoma
73. Development of Selective Cyclin-Dependent Kinase 4 Inhibitors for Antineoplastic Therapies
74. Discovery and Biological Evaluation of a Series of Pyrrolo[2,3-b]pyrazines as Novel FGFR Inhibitors
75. Discovery and Biological Evaluation of a Series of Pyrrolo[2,3-b]pyrazines as Novel FGFR Inhibitors
76. A one-pot synthesis of omarigliptin and its analogues through stabilized beta-amino ketone intermediate
77. Stereoselective and Regioselective Preparation ofC-Pentopyranosides and Formal Synthesis of Omarigliptin
78. 1,2-trans-1-Dihydroxyboryl benzyl S-glycoside as glycosyl donor
79. Identification of a new series of potent diphenol HSP90 inhibitors by fragment merging and structure-based optimization
80. Design, Synthesis and Biological Evaluation of 6-(2,6-Dichloro-3,5-dimethoxyphenyl)-4-substituted-1H-indazoles as Potent Fibroblast Growth Factor Receptor Inhibitors
81. Molecular regulation of apoptotic machinery and lipid metabolism by mTORC1/mTORC2 dual inhibitors in preclinical models of HER2+/PIK3CAmut breast cancer
82. ChemInform Abstract: Formation of 1,3‐Diazocine by Palladium Catalyzed C—H Arylation.
83. Tetrahydroisoquinolines as novel histone deacetylase inhibitors for treatment of cancer
84. CCLab—a multi-objective genetic algorithm based combinatorial library design software and an application for histone deacetylase inhibitor design
85. ChemInform Abstract: Ga(OTf)3‐Promoted Synthesis of Functionalized 2‐Carbonyl‐imidazo[1,2‐a]pyridines Derived from Ethyl α‐Benzotriazolyl‐α‐morpholinoacetate.
86. FS-93, an Hsp90 inhibitor, induces G2/M arrest and apoptosis via the degradation of client proteins in oncogene addicted and derived resistant cancer cells
87. ChemInform Abstract: An Efficient Synthesis of Novel Dibenzoxdiazepine-Fused Heterocycles Through a Multicomponent Reaction.
88. Design and Optimization of a Series of 1-Sulfonylpyrazolo[4,3-b]pyridines as Selective c-Met Inhibitors
89. Fragment-Based Drug Discovery of 2-Thiazolidinones as BRD4 Inhibitors: 2. Structure-Based Optimization
90. Multi-substituted 8-aminoimidazo[1,2-a]pyrazines by Groebke–Blackburn–Bienaymé reaction and their Hsp90 inhibitory activity
91. Ga(OTf)3-promoted synthesis of functionalized 2-carbonyl-imidazo[1,2-a]pyridines derived from ethyl α-benzotriazolyl-α-morpholinoacetate
92. A Chemical Tuned Strategy to Develop Novel Irreversible EGFR-TK Inhibitors with Improved Safety and Pharmacokinetic Profiles
93. Discovery and Optimization of 4,5-Diarylisoxazoles as Potent Dual Inhibitors of Pyruvate Dehydrogenase Kinase and Heat Shock Protein 90
94. Potent and novel 11β-HSD1 inhibitors identified from shape and docking based virtual screening
95. Stereoselective and Regioselective Preparation of C-Pentopyranosides and Formal Synthesis of Omarigliptin.
96. Highly Stereoselective Nucleophilic Addition of Difluoromethyl-2-pyridyl Sulfone to Sugar Lactones and Efficient Synthesis of Fluorinated 2-Ketoses
97. Neoglycopeptide Synthesis by Suzuki-Miyaura Couplings between Glycosyl Aryl Boronic Acids and Iodopeptides
98. A Novel Strategy for Preparing Glycopeptide Molecular Probe Using Fluorous Technology
99. Mechanism of the All-α to All-β Conformational Transition of RfaH-CTD: Molecular Dynamics Simulation and Markov State Model
100. Direct Glycosylation of Bioactive Small Molecules with Glycosyl Iodide and Strained Olefin as Acid Scavenger
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