383 results on '"Rautio, Jarkko"'
Search Results
52. Prodrug Strategies in Drug Design
53. Enzyme-Activated Prodrug Strategies for Targeted Drug Action
54. Synthesis and In Vitro Evaluation of Aminoacyloxyalkyl Esters of 2-(6-methoxy-2-naphthyl)propionic Acid as Novel Naproxen Prodrugs for Dermal Drug Delivery
55. Amino acid prodrugs for oral delivery: challenges and opportunities
56. Addressing the Biochemical Foundations of a Glucose-Based “Trojan Horse”-Strategy to Boron Neutron Capture Therapy: From Chemical Synthesis to In Vitro Assessment
57. Anti-bacterial activity of inorganic nanomaterials and their antimicrobial peptide conjugates against resistant and non-resistant pathogens
58. Prodrug Approach for Posterior Eye Drug Delivery: Synthesis of Novel Ganciclovir Prodrugs and in Vitro Screening with Cassette Dosing
59. Tyrosine–Chlorambucil Conjugates Facilitate Cellular Uptake through L-Type Amino Acid Transporter 1 (LAT1) in Human Breast Cancer Cell Line MCF-7
60. Brain uptake of ketoprofen–lysine prodrug in rats
61. Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–6
62. Role of L-Type Amino Acid Transporter 1 (LAT1) for the Selective Cytotoxicity of Sesamol in Human Melanoma Cells
63. Design and Pharmaceutical Applications of Prodrugs
64. Synthesis, in vitro and in vivo characterization of novel ethyl dioxy phosphate prodrug of propofol
65. Diclofenac readily penetrates the cerebrospinal fluid in children
66. Enhanced brain drug delivery and targeting: an examination of the drug analogs and prodrugs of small molecules that utilize either large neutral amino acid or glucose transporters of the BBB in their brain penetration
67. Inefficient central nervous system delivery limits the use of ibuprofen in neurodegenerative diseases
68. Synthesis and antileishmanial activity of novel buparvaquone oxime derivatives
69. Design, synthesis and in vitro evaluation of novel water-soluble prodrugs of buparvaquone
70. Secondary carbamate linker can facilitate the sustained release of dopamine from brain-targeted prodrug
71. Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–5
72. Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-2Molecules
73. Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–4
74. Discovery of polar spirocyclic orally bioavailable urea inhibitors of soluble epoxide hydrolase
75. Synthesis, Stability and In Vitro Dermal Evaluation of Aminocarbonyloxymethyl Esters as Prodrugs of Carboxylic Acid Agents
76. Exploring the Biochemical Foundations of a Successful GLUT1-Targeting Strategy to BNCT: Chemical Synthesis and In Vitro Evaluation of the Entire Positional Isomer Library of ortho-Carboranylmethyl-Bearing Glucoconjugates.
77. Erratum to: Design, Synthesis and Brain Uptake of LAT1-Targeted Amino Acid Prodrugs of Dopamine
78. Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3
79. Structural properties for selective and efficient l-type amino acid transporter 1 (LAT1) mediated cellular uptake
80. The expanding role of prodrugs in contemporary drug design and development
81. Exploring the Biochemical Foundations of a Successful GLUT1-Targeting Strategy to BNCT: Chemical Synthesis and In VitroEvaluation of the Entire Positional Isomer Library of ortho-Carboranylmethyl-Bearing Glucoconjugates
82. Glutathione-S-transferase selective release of metformin from its sulfonamide prodrug
83. Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-2.
84. Evaluation of Novel Imidazotetrazine Analogues Designed to Overcome Temozolomide Resistance and Glioblastoma Regrowth
85. Brain Pharmacokinetics of Ganciclovir in Rats with Orthotopic BT4C Glioma
86. Aminocarbonyloxymethyl ester prodrugs of flufenamic acid and diclofenac
87. Quantitative Insight into the Design of Compounds Recognized by the L‐Type Amino Acid Transporter 1 (LAT1)
88. Potenciais Pró-Fármacos do Ácido Flufenâmico
89. Inhibitors of LRRK2 Kinase Activity To Probe the Treatment Option in Parkinson’s Disease
90. Design, Synthesis, and Evaluation of Novel Cyclic Phosphates of 5-Aminosalicylic Acid as Cytochrome P450-Activated Prodrugs
91. Prodrugs - An Efficient Way to Breach Delivery and Targeting Barriers
92. Large Amino Acid Transporter 1 (LAT1) Prodrugs of Valproic Acid: New Prodrug Design Ideas for Central Nervous System Delivery
93. Prodrugs—from Serendipity to Rational Design
94. Design, synthesis and in vitro/in vivo evaluation of orally bioavailable prodrugs of a catechol-O-methyltransferase inhibitor
95. Design and Pharmaceutical Applications of Prodrugs
96. The First Bioreversible Prodrug of Metformin with Improved Lipophilicity and Enhanced Intestinal Absorption
97. Glucose Promoiety Enables Glucose Transporter Mediated Brain Uptake of Ketoprofen and Indomethacin Prodrugs in Rats
98. Cytochrome P450-Activated Prodrugs: Targeted Drug Delivery
99. Prodrugs: design and clinical applications
100. Large Neutral Amino Acid Transporter Enables Brain Drug Delivery via Prodrugs
Catalog
Books, media, physical & digital resources
Discovery Service for Jio Institute Digital Library
For full access to our library's resources, please sign in.