116 results on '"Portoghese, Philip S."'
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2. Opioid-Induced Tolerance and Dependence in Mice Is Modulated by the Distance between Pharmacophores in a Bivalent Ligand Series
3. A Heterodimer-Selective Agonist Shows in vivo Relevance of G Protein-Coupled Receptor Dimers
4. Bivalent ligand that activates mu opioid receptor and antagonizes mGluR5 receptor reduces neuropathic pain in mice
5. A bivalent compound targeting CCR5 and the mu opioid receptor treats inflammatory arthritis pain in mice without inducing pharmacologic tolerance
6. Ligands that interact with putative MOR-mGluR5 heteromer in mice with inflammatory pain produce potent antinociception
7. N-naphthoyl-ß-naltrexamine (NNTA), a highly selective and potent activator of μ/κ-opioid heteromers
8. Naloxone Acts as a Potent Analgesic in Transgenic Mouse Models of Sickle Cell Anemia
9. Targeting putative mu opioid/metabotropic glutamate receptor-5 heteromers produces potent antinociception in a chronic murine bone cancer model
10. Consequences of opioid receptor mutation on actions of univalent and bivalent kappa and delta ligands
11. Absence of conditioned place preference or reinstatement with bivalent ligands containing mu-opioid receptor agonist and delta-opioid receptor antagonist pharmacophores
12. Effects of κ-opioid receptor ligands on intracranial self-stimulation in rats
13. Opioid-induced tolerance and dependence in mice is modulated by the distance between pharmacophores in a bivalent ligand series
14. Specific cross-linking of Lys233 and Cys235 in the mu opioid receptor by a reporter affinity label
15. Kappa opioid antagonist effects of the novel kappa antagonist 5′-guanidinonaltrindole (GNTI) in an assay of schedule-controlled behavior in rhesus monkeys
16. GRAS flavoring substances 21: the 21st publication by the Expert Panel of the Flavor and Extract Manufacturers Association on recent progress in the consideration of flavoring ingredients generally recognized as safe under the Food Additives Amendment
17. The δ2-opioid receptor antagonist naltriben reduces motivated responding for ethanol
18. Criteria for the safety evaluation of flavoring substances: The Expert Panel of the Flavor and Extract Manufacturers Association
19. Application of the message-address concept to the docking of naltrexone and selective naltrexone-derived opioid antagonists into opioid receptor models
20. Identification of Helical Packing Motifs Common to Bacteriorhodopsin and G Protein-Coupled Receptors
21. Boron tribromide-catalyzed rearrangement of 7,7-diphenylhydromorphone to 6,7-diphenylmorphine: a novel conversion of ketones to allylic alcohols
22. The FEMA GRAS assessment of cinnamyl derivatives used as flavor ingredients
23. Chloroxymorphamine, an Opioid Receptor Site-Directed Alkylating Agent Having Narcotic Agonist Activity
24. Effect of opioid receptor ligands on the μ-S196A knock-in and μ knockout mouse vas deferens
25. Identity of the putative δ1-opioid receptor as a δ–κ heteromer in the mouse spinal cord
26. In Memory of Professor Hualiang Jiang.
27. Opiate dienes as dienophiles in the Diels-Alder reaction with 1-cyano-o-quinodimethane
28. The bivalent ligand, MMG22, reduces neuropathic pain after nerve injury without the side effects of traditional opioids.
29. Monophenylation of morphinan-6-ones with diphenyliodonium iodide
30. Endomorphin-1 potentiates HIV-1 expression in human brain cell cultures: implication of an atypical μ-opoid receptor
31. Stereochemistry and innate immune recognition: (+)-norbinaltorphimine targets myeloid differentiation protein 2 and inhibits toll-like receptor 4 signaling.
32. Combined Glia Inhibition and Opioid Receptor Agonism Afford Highly Potent Analgesics without Tolerance.
33. Bivalent ligand MCC22 potently attenuates nociception in a murine model of sickle cell disease.
34. Modulation of musculoskeletal hyperalgesia by brown adipose tissue activity in mice.
35. Stereospecific synthesis of pseudocodeine: (2,3)-sigmatropic rearrangement using selenium intermediates
36. Putative Kappa Opioid HeteromersAs Targets for Developing Analgesics Free of Adverse Effects.
37. BivalentLigands That Target μ Opioid (MOP)and Cannabinoid1 (CB1) Receptors Are Potent AnalgesicsDevoid of Tolerance.
38. Reduced Antinociceptionof Opioids in Rats and Mice by Vaccination with Immunogens ContainingOxycodone and Hydrocodone Haptens.
39. Opioid Activity of SpinallySelective Analogues of N-Naphthoyl-β-naltrexaminein HEK-293 Cells and Mice.
40. MDAN-21: A Bivalent Opioid Ligand Containing mu-Agonist and Delta-Antagonist Pharmacophores and Its Effects in Rhesus Monkeys.
41. N-naphthoyl-β-naltrexamine (NNTA), a highly selective and potent activator of μ/κ-opioid heteromers.
42. Modulation of Cell Surface Expression of Nonactivated Cholecystokinin Receptors Using Bivalent Ligand-Induced Internalization.
43. Synthesis and 124I-labeling of m-iodophenylpyrrolomorphinan as a potential PET imaging agent for delta opioid (DOP) receptors.
44. N1'-( p-[18F]Fluorobenzyl)naltrindole ( p-[18F]BNTI) as a potential PET imaging agent for DOP receptors.
45. Specific Cross-Linking of Lys233 and Cys235 in the Mu Opioid Receptor by a Reporter Affinity Label.
46. The δ[sub 2] -opioid receptor antagonist naltriben reduces motivated responding for ethanol.
47. Synthesis and physico-chemical properties of (R, S)-6-ditrideuteriomethylamino-4,4-diphenylheptan-3-one hydrochloride (methadone-d6).
48. Synthesis of [3H]DIPPA: A potent irreversible antagonist selective for the κ opioid receptor.
49. Molecular modeling of the conformational and sodium ion binding properties of the oligosaccharide component of ganglioside GM1.
50. Identity of the putative δ1-opioid receptor as a δ–κ heteromer in the mouse spinal cord
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