129 results on '"Ghosh, Arun K"'
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2. Asymmetric 1,2‐Carbamoyl Rearrangement of Lithiated Chiral Oxazolidine Carbamates and Diastereoselective Synthesis of α‐Hydroxy Amides
3. Design, Synthesis and X‐ray Structural Studies of Potent HIV‐1 Protease Inhibitors Containing C‐4 Substituted Tricyclic Hexahydro‐furofuran derivatives as P2 ligands
4. Aspartic Acid Proteases as Therapeutic Targets
5. Drug Development and Medicinal Chemistry Efforts toward SARS‐Coronavirus and Covid‐19 Therapeutics
6. Potent HIV‐1 Protease Inhibitors Containing Carboxylic and Boronic Acids: Effect on Enzyme Inhibition and Antiviral Activity and Protein‐Ligand X‐ray Structural Studies
7. Cover Feature: Highly Selective and Potent Human β-Secretase 2 (BACE2) Inhibitors against Type 2 Diabetes: Design, Synthesis, X-ray Structure and Structure-Activity Relationship Studies (ChemMedChem 5/2019)
8. Highly Selective and Potent Human β‐Secretase 2 (BACE2) Inhibitors against Type 2 Diabetes: Design, Synthesis, X‐ray Structure and Structure–Activity Relationship Studies
9. The Curtius Rearrangement: Applications in Modern Drug Discovery and Medicinal Chemistry
10. Nature Inspired Molecular Design: Stereoselective Synthesis of Bicyclic and Polycyclic Ethers for Potent HIV-1 Protease Inhibitors
11. Front Cover: Design of Highly Potent, Dual-Acting and Central-Nervous-System-Penetrating HIV-1 Protease Inhibitors with Excellent Potency against Multidrug-Resistant HIV-1 Variants (ChemMedChem 8/2018)
12. Design of Highly Potent, Dual‐Acting and Central‐Nervous‐System‐Penetrating HIV‐1 Protease Inhibitors with Excellent Potency against Multidrug‐Resistant HIV‐1 Variants
13. Enantioselective Syntheses of (-)-Alloyohimbane and (-)-Yohimbane by an Efficient Enzymatic Desymmetrization Process
14. ChemInform Abstract: Stereoselective Synthesis of Substituted Oxocene Cores by Lewis Acid Promoted Cyclization.
15. Development of an efficient structure‐based drug discovery platform for BACE1 Inhibitors for the treatment of Alzheimer's Disease
16. Prospects of β‐Secretase Inhibitors for the Treatment of Alzheimer’s Disease
17. ChemInform Abstract: A Convergent Synthesis of Carbocyclic Sinefungin (Ia) and Its C-5 Epimer (Ib).
18. ChemInform Abstract: FeCl3-Catalyzed Tandem Prins and Friedel-Crafts Cyclization: A Highly Diastereoselective Route to Polycyclic Ring Structures.
19. Design of gem‐Difluoro‐bis‐Tetrahydrofuran as P2 Ligand for HIV‐1 Protease Inhibitors to Improve Brain Penetration: Synthesis, X‐ray Studies, and Biological Evaluation
20. A Convergent Synthesis of Carbocyclic Sinefungin and its C-5 Epimer
21. ChemInform Abstract: An Intramolecular Cascade Cyclization of 2‐Aryl Indoles: Efficient Methods for the Construction of 2,3‐Functionalized Indolines and 3‐Indolinones.
22. Proteasome Inhibitors for the Treatment of Relapsed Multiple Myeloma: Design and Discovery of Bortezomib and Carfilzomib
23. Structure‐Based Design of Drugs and Other Bioactive Molecules
24. ChemInform Abstract: Enantioselective Total Synthesis of Macrolide (+)-Neopeltolide (I).
25. ChemInform Abstract: Enantioselective Syntheses of FR901464 (Ib) and Spliceostatin A (Ia): Potent Inhibitors of Spliceosome.
26. ChemInform Abstract: Bifunctional Cinchona Alkaloid Squaramide Catalyzed Highly Enantioselective Aza‐Michael Addition of Indolines to α,β‐Unsaturated Ketones.
27. ChemInform Abstract: Enantioselective Synthesis of Spiro[cyclohexane-1,3′-indolin]-2′-ones Containing Multiple Stereocenters via Organocatalytic Michael/Aldol Cascade Reactions.
28. Synergistic Inhibitor Binding to the Papain-Like Protease of Human SARS Coronavirus: Mechanistic and Inhibitor Design Implications
29. Metabolism‐Directed Structure Optimization of Benzimidazole‐Based F. Tularensis Enoyl‐Reductase (FabI) Inhibitors
30. ChemInform Abstract: Diastereoselective Synthesis of Substituted Tetrahydropyrans by Copper(II)—Bisphosphine‐Catalyzed Olefin Migration and Prins Cyclization.
31. Candida albicanssecreted aspartic proteases 4–6 induce apoptosis of epithelial cells by a novel Trojan horse mechanism
32. ChemInform Abstract: A Tandem Olefin Migration and Prins Cyclization Using Cu(OTf)2-Bisphosphine Complexes: An Improved Synthesis of Functionalized Tetrahydropyrans.
33. ChemInform Abstract: Expedient Synthesis of α-Substituted Fluoroethenes.
34. ChemInform Abstract: Synthesis of Functionalized 4-Methylenetetrahydropyrans by Oxidative Activation of Cinnamyl or Benzyl Ethers.
35. ChemInform Abstract: TiCl4‐Promoted Tandem Carbonyl or Imine Addition and Friedel—Crafts Cyclization: Synthesis of Benzo‐Fused Oxabicyclooctanes and Nonanes.
36. Total Synthesis of Potent Antitumor Macrolide (–)‐Zampanolide: An Oxidative Intramolecular Cyclization‐Based Strategy
37. ChemInform Abstract: Enhancing Protein Backbone Binding — A Fruitful Concept for Combating Drug‐Resistant HIV.
38. Enhancing Protein Backbone Binding-A Fruitful Concept for Combating Drug-Resistant HIV
39. Verstärkung der Bindung an das Proteinrückgrat - ein fruchtbares Konzept gegen die Arzneimittelresistenz von HIV
40. Critical differences in HIV-1 and HIV-2 protease specificity for clinical inhibitors
41. ChemInform Abstract: Cu(II)-Catalyzed Olefin Migration and Prins Cyclization: Highly Diastereoselective Synthesis of Substituted Tetrahydropyrans.
42. Developing β-secretase inhibitors for treatment of Alzheimer’s disease
43. ChemInform Abstract: Capturing the Essence of Organic Synthesis: From Bioactive Natural Products to Designed Molecules in Today′s Medicine
44. β‐Secretase inhibitor GRL‐8234 rescues age‐related cognitive decline in APP transgenic mice
45. Cover Picture: Probing Multidrug-Resistance and Protein-Ligand Interactions with Oxatricyclic Designed Ligands in HIV-1 Protease Inhibitors (ChemMedChem 11/2010)
46. ChemInform Abstract: Enantioselective Syntheses of the Proposed Structures of Cytotoxic Macrolides Iriomoteolide‐1a (I) and ‐1b (II).
47. Probing Multidrug-Resistance and Protein-Ligand Interactions with Oxatricyclic Designed Ligands in HIV-1 Protease Inhibitors
48. TheFDAApprovedHIV‐1 Protease Inhibitors for Treatment ofHIV/AIDS
49. The Discovery of β‐Secretase and Development toward a Clinical Inhibitor for AD: An Exciting Academic Collaboration
50. ChemInform Abstract: Bis(oxazoline) Derived Cationic Aqua Complexes: Highly Effective Catalysts for Enantioselective Diels-Alder Reactions.
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