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6 results on '"Lipford, J Russell"'

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1. Mercapturate pathway metabolites of sotorasib, a covalent inhibitor of KRASG12C, are associated with renal toxicity in the Sprague Dawley rat

2. Discovery of imidazopyridazines as potent Pim-1/2 kinase inhibitors

3. The discovery and optimization of aminooxadiazoles as potent Pim kinase inhibitors

4. The discovery of novel 3-(pyrazin-2-yl)-1H-indazoles as potent pan-Pim kinase inhibitors

5. Discovery of 5-(1H-indol-5-yl)-1,3,4-thiadiazol-2-amines as potent PIM inhibitors

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