8 results on '"Kosaka, Takatoshi"'
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2. trans -(3 S ,4 S )-Disubstituted pyrrolidines as inhibitors of the human aspartyl protease renin. Part I: Prime site exploration using an amino linker
3. Novel ROCK inhibitors for the treatment of pulmonary arterial hypertension
4. Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-Cyanopyrimidines. Part 2
5. 4-Amino-2-cyanopyrimidines: Novel scaffold for nonpeptidic cathepsin S inhibitors
6. Discovery of selective and nonpeptidic cathepsin S inhibitors
7. Enantioselective synthesis of neoambrosin, parthenin, and dihydroisoparthenin
8. A novel series of highly potent 5-lipoxygenase inhibitors; 2-aryldienylbenzoxazoles
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