156 results on '"Pieroni, Marco"'
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2. Public governance: the influence of corporate governance in strengthening AGU'S strategic management/Governanca publica: a influencia da governanca corporative no fortalecimento da gestao estrategica da AGU/Gobierno publico: la influencia del gobierno corporativo en el fortalecimiento de la gestion estrategica de la AGU
3. Expanding the knowledge around antitubercular 5-(2-aminothiazol-4-yl)isoxazole-3-carboxamides: Hit–to–lead optimization and release of a novel antitubercular chemotype via scaffold derivatization
4. Governança pública: a influência da governança corporativa no fortalecimento da gestão estratégica da AGU.
5. Exploring the chemical space around N-(5-nitrothiazol-2-yl)-1,2,3-thiadiazole-4-carboxamide, a hit compound with serine acetyltransferase (SAT) inhibitory properties
6. Towards the sustainable discovery and development of new antibiotics
7. Chemical Probes to Investigate Central Nervous System Disorders: Design, Synthesis and Mechanism of Action of a Potent Human Serine Racemase Inhibitor.
8. Antituberculosis agents: Beyond medicinal chemistry rules
9. Modulation of bacterial metabolism by the microenvironment controls MAIT cell stimulation
10. A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin
11. Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design
12. Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A
13. Identification of Human Alanine–Glyoxylate Aminotransferase Ligands as Pharmacological Chaperones for Variants Associated with Primary Hyperoxaluria Type 1
14. Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria
15. Crystal structure of Aspergillus fumigatusAroH, an aromatic amino acid aminotransferase
16. Roadmap towards the sustainable discovery and development of new antibiotics
17. A Competitive O-Acetylserine Sulfhydrylase Inhibitor Modulates the Formation of Cysteine Synthase Complex
18. Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants
19. Investigational Studies on a Hit Compound Cyclopropane–Carboxylic Acid Derivative Targeting O-Acetylserine Sulfhydrylase as a Colistin Adjuvant
20. Aspergillus fumigatus tryptophan metabolic route differently affects host immunity
21. Nitric oxide-releasing cyclodextrins as biodegradable antibacterial scaffolds: a patent evaluation of US2019343869(A1)
22. 2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry
23. Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor
24. Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: implications for Primary Hyperoxaluria type 1
25. Crystal structure of Aspergillus fumigatusAroH, an aromatic amino acid aminotransferase.
26. Challenging the drug-likeness dogma for new drug discovery in Tuberculosis
27. Sodium Hyaluronate Nanocomposite Respirable Microparticles to Tackle Antibiotic Resistance with Potential Application in Treatment of Mycobacterial Pulmonary Infections
28. Cycloserine enantiomers are reversible inhibitors of human alanine: glyoxylate aminotransferase: implications for Primary Hyperoxaluria type 1.
29. Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms.
30. Biochemical Characterization of Aspergillus fumigatus AroH, a Putative Aromatic Amino Acid Aminotransferase
31. Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms
32. In vitro Digestion of Zingiber officinale Extract and Evaluation of Stability as a First Step to Determine its Bioaccesibility
33. Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting Mycobacterium tuberculosis energetics
34. Challenging the Drug-Likeness Dogma for New Drug Discovery in Tuberculosis
35. Efflux Activity Differentially Modulates the Levels of Isoniazid and Rifampicin Resistance among Multidrug Resistant and Monoresistant Mycobacterium tuberculosis Strains
36. Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets
37. Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design
38. Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases
39. Substituted N-Phenyl-5-(2-(phenylamino)thiazol-4-yl)isoxazole-3-carboxamides Are Valuable Antitubercular Candidates that Evade Innate Efflux Machinery
40. Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure–Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents
41. Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary Diseases
42. An Experimental Model for the Rapid Screening of Compounds with Potential Use Against Mycobacteria
43. Cover Picture: Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches (ChemMedChem 17/2016)
44. Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation ofO-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR
45. Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches
46. Rational Design, Synthesis, and Preliminary Structure–Activity Relationships of α-Substituted-2-Phenylcyclopropane Carboxylic Acids as Inhibitors of Salmonella typhimurium O-Acetylserine Sulfhydrylase
47. Mutation of Rv2887 , a marR -Like Gene, Confers Mycobacterium tuberculosis Resistance to an Imidazopyridine-Based Agent
48. Rational Design and Synthesis of Thioridazine Analogues as Enhancers of the Antituberculosis Therapy
49. Cyclopropane derivatives as potential human serine racemase inhibitors: unveiling novel insights into a difficult target
50. Synthesis of 7-Desmethyl Analogs of (+)- and (−)-Huperzine A
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