132 results on '"Cerra, Bruno"'
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2. Chemical exploration of TGR5 functional hot-spots: Synthesis and structure-activity relationships of C7- and C23-Substituted cholic acid derivatives
3. Development of 3α,7α-dihydroxy-6α-ethyl-24-nor-5β-cholan-23-sulfate sodium salt (INT-767): Process optimization, synthesis and characterization of metabolites
4. Patented Farnesoid X receptor modulators: a review (2019 – present)
5. Future medicinal chemists experience flow chemistry: optimization by experimental design of the limiting synthetic step to the antifungal drug econazole nitrate
6. Continuous Flow Synthesis of the PARP-1/2 Inhibitor HYDAMTIQ: Synthetic Strategy, Optimization, and Green Metrics Evaluation.
7. Integrating experimental and computational techniques to study chromatographic enantioresolutions of chiral tetrahydroindazole derivatives
8. Continuous Flow Synthesis of the PARP-1/2 Inhibitor HYDAMTIQ: Synthetic Strategy, Optimization, and Green Metrics Evaluation
9. Synthesis, physicochemical properties, and biological activity of bile acids 3-glucuronides: Novel insights into bile acid signalling and detoxification
10. Merging Continuous Flow Technology, Photochemistry and Biocatalysis to Streamline Steroid Synthesis
11. Multi-Gram Scale Synthesis and Characterization of Mometasone Furoate EP Impurity C.
12. Integrated Systems for Continuous Synthesis and Biological Screenings
13. Turning a Tumor Microenvironment Pitfall into Opportunity: Discovery of Benzamidoxime as PD-L1 Ligand with pH-Dependent Potency
14. Multicomponent and Metal‐Free Diels–Alder/Aromatization Approach to the Stereospecific Synthesis of E‐(Hetero)Stilbenes and Diarylacetylenes.
15. Isocyanide chemistry enabled by continuous flow technology
16. Isocyanide Chemistry Enabled by Continuous Flow Technology
17. Combining molecular modeling approaches to establish the chromatographic enantiomer elution order in the absence of pure enantiomeric standards: A study case with two tetracyclic quinolines
18. The Systems Biology of Transporters - Targeting the Regulatory System for Transporters (FXR/RXR)
19. Concepts and Optimization Strategies of Experimental Design in Continuous-Flow Processing
20. Integrated Systems for Continuous Synthesis and Biological Screenings
21. Domino synthesis of 5-aminoimidazoles from Strecker multicomponent adducts via ytterbium-promoted isocyanide insertion/5-exo-dig cyclization
22. Development of 3α,7α-Dihydroxy-6α-ethyl-24-nor-5b-Cholan-23-Sulfate Sodium Salt (INT-767): Process Optimization, Synthesis and Characterization of Metabolites
23. The Stone Guest: How Does pH Affect Binding Properties of PD‐1/PD‐L1 Inhibitors?
24. Garcinoic Acid Is a Natural and Selective Agonist of Pregnane X Receptor
25. The Medicinal Chemistry in the Era of Machines and Automation: Recent Advances in Continuous Flow Technology
26. Enantioselective HPLC Analysis to Assist the Chemical Exploration of Chiral Imidazolines
27. A streamlined synthesis of the neurosteroid 3β-methoxypregnenolone assisted by a statistical experimental design and automation
28. Garcinoic Acid Is a Natural and Selective Agonist of Pregnane X Receptor
29. Optimisation by Design of Experiment of Benzimidazol-2-One Synthesis under Flow Conditions
30. In-Flow Flash Nanoprecipitation of Size-Controlled D-Leucine Nanoparticles for Spray-Drying Formulations
31. Flow nanoprecipitation of size-controlled d-leucine nanoparticles for spray-drying formulations
32. Exploiting Chemical Toolboxes for the Expedited Generation of Tetracyclic Quinolines as a Novel Class of PXR Agonists
33. BF3·Et2O-Promoted Decomposition of Cyclic α-Diazo-β-Hydroxy Ketones: Novel Insights into Mechanistic Aspects
34. The Stone Guest: How Does pH Affect Binding Properties of PD‐1/PD‐L1 Inhibitors?
35. 9. The Systems Biology of Transporters – Targeting the Regulatory System for Transporters (FXR/RXR)
36. Synthesis of hydroxy lactones by selenium-mediated oxidation/cyclization of alkenoic acids under eco-flow conditions
37. Continuous Flow Synthesis of 16-Dehydropregnenolone Acetate, a Key Synthon for Natural Steroids and Drugs
38. Binding Mode and Structure-Activity Relationships of ITE as an Aryl Hydrocarbon Receptor (AhR) Agonist
39. Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms
40. Front Cover Picture: Merging Continuous Flow Technology, Photochemistry and Biocatalysis to Streamline Steroid Synthesis (Adv. Synth. Catal. 23/2023).
41. Speeding up Early Phases of Drug Discovery: DoE-Driven Synthetic Optimization of Chemical Processes in Flow Systems
42. ATYPICAL BILE ACIDS AS CHEMICAL PROBES FOR DIAGNOSIS AND THERAPHY MONITORING OF PROGRESSIVE CHOLESTATIC LIVER DISEASE IN HSD3B7 PATIENTS
43. IDENTIFICATION OF A NOVEL CLASS OF PREGNANE X RECEPTOR (PXR) LIGANDS: FLOW SYNTHESIS AND PRELIMINARY BIOLOGICAL ACTIVITY OF TETRAHYDROQUINOLINES
44. Selected cholesterol biosynthesis inhibitors produce accumulation of the intermediate FF-MAS that targets nucleus and activates LXRα in HepG2 cells
45. Selective continuous flow synthesis of hydroxy lactones from alkenoic acids
46. Exploiting Chemical Toolboxes for the Expedited Generation of Tetracyclic Quinolines as a Novel Class of PXR Agonists.
47. Integrating multicomponent flow synthesis and computational approaches for the generation of a tetrahydroquinoline compound based library
48. First Total Synthesis of Piperenol B and Configuration Revision of the Enantiomers Piperenol B and Uvarirufol A
49. Bile Acid Derivatives as Ligands of the Farnesoid X Receptor: Molecular Determinants for Bile Acid Binding and Receptor Modulation
50. Beyond Bile Acids: Targeting Farnesoid X Receptor (FXR) with Natural and Synthetic Ligands
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