15 results on '"Shen, Jingkang"'
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2. Fragment-based drug discovery of triazole inhibitors to block PDEδ-RAS protein-protein interaction
3. Discovery and optimization of a series of 3-substituted indazole derivatives as multi-target kinase inhibitors for the treatment of lung squamous cell carcinoma
4. Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups
5. Discovery of novel high potent and cellular active ADC type PTP1B inhibitors with selectivity over TC-PTP via modification interacting with C site
6. Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor
7. Discovery of novel, high potent, ABC type PTP1B inhibitors with TCPTP selectivity and cellular activity
8. Discovery of potent N-(isoxazol-5-yl)amides as HSP90 inhibitors
9. Discovery of pyrazole as C-terminus of selective BACE1 inhibitors
10. Design, synthesis and SAR of piperidyl-oxadiazoles as 11β-hydroxysteroid dehydrogenase 1 inhibitors
11. Asymmetric synthesis and biological evaluation of N-cyclohexyl-4-[1-(2,4-dichlorophenyl)-1-(p-tolyl)methyl]piperazine-1-carboxamide as hCB1 receptor antagonists
12. Discovery of benzhydrylpiperazine derivatives as CB 1 receptor inverse agonists via privileged structure-based approach
13. Discovery of novel 2-phenyl-imidazo[1,2-a]pyridine analogues targeting tubulin polymerization as antiproliferative agents
14. Discovery of benzhydrylpiperazine derivatives as CB1 receptor inverse agonists via privileged structure-based approach
15. Discovery of benzhydrylpiperazine derivatives as CB1 receptor inverse agonists via privileged structure-based approach
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