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2. Design and Synthesis of Novel 2-Acetamido, 6-Carboxamide Substituted Benzothiazoles as Potential BRAFV600E Inhibitors - In vitro Evaluation of their Antiproliferative Activity.
3. Corrigendum: Covalent Complex of DNA and Bacterial Topoisomerase: Implications in Antibacterial Drug Development.
4. Diastereoselective Cascade Double Michael Addition to Access Bridged Coumarins, Oxindoles and Spirooxindoles: A Sustainable Strategy for Synthesis of Anticancer Molecules.
5. 4-Aza Cyclopentenone Prostaglandin Analogues: Synthesis and NF-κB Inhibitory Activities.
6. Design, Synthesis and Biological Evaluation of Novel Anticancer Amidinourea Analogues via Unexpected 1,3,5‐Triazin‐2‐one Ring Opening.
7. C7‐Halomethylene/methyl‐C3‐thiophenyl‐spirocyclic‐β‐lactams: Synthesis, X‐ray Analysis, Antimicrobial Evaluation, Cytotoxicity Profile and Molecular Docking Interactions.
8. Evaluation of Rhodanine Indolinones as AANAT Inhibitors.
9. Structural Optimization of Antimycobacterial Azaaurones Towards Improved Solubility and Metabolic Stability.
10. Terpene‐Functionalized Fluoroquinolones as Potential Antimicrobials: Synthesis and Properties.
11. Synergistic and Additive Effects of Menadione in Combination with Antibiotics on Multidrug‐Resistant Staphylococcus aureus: Insights from Structure‐Function Analysis of Naphthoquinones.
12. Targeting EPHA2 with Kinase Inhibitors in Colorectal Cancer.
13. Protein‐Porphyrin Complex Photosensitizers for Anticancer and Antimicrobial Photodynamic Therapies.
14. Moving out of CF3‐Land: Synthesis, Receptor Affinity, and in silico Studies of NK1 Receptor Ligands Containing a Pentafluorosulfanyl (SF5) Group.
15. Development of Photoswitchable Tethered Ligands that Target the μ‐Opioid Receptor.
16. Cellular Effects of Cationic Copper(II) Schiff Base Complexes: Anti-Inflammatory and Antiproliferative Properties.
17. 5‐Substituted Uridines with Activity against Gram‐Positive Bacteria.
18. Exploration of the Pharmacophore for Cytoskeletal Targeting Ruthenium Polypyridyl Complexes.
19. Design and Synthesis of Highly Potent and Specific ABHD6 Inhibitors.
20. Screening Campaign and Docking Investigations in Identifying New Hit Compounds as Inhibitors of Human Carbonic Anhydrases Expressed In Tumour Cells.
21. Zwitterionic Polymer: A New Paradigm for Protein Conjugation beyond PEG.
22. Design, Synthesis of (±)‐Millpuline A, and Biological Evaluation for the Lung Cell Protective Effects through SRC.
23. Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors.
24. RNA‐Selective Small‐Molecule Ligands: Recent Advances in Live‐Cell Imaging and Drug Discovery.
25. Lysyl Oxidases as Targets for Cancer Therapy and Diagnostic Imaging.
26. Total Synthesis and Biological Investigation of Mindapyrroles A and B.
27. Insights into the Pharmacological Activity of the Imidazo−Pyrazole Scaffold.
28. Cell Penetrating Peptides: Classification, Mechanisms, Methods of Study, and Applications.
29. A Patent Review on SARS Coronavirus Papain‐Like Protease (PLpro) Inhibitors.
30. A Study of the Activity of Adamantyl Amines against Mutant Influenza A M2 Channels Identified a Polycyclic Cage Amine Triple Blocker, Explored by Molecular Dynamics Simulations and Solid‐State NMR**.
31. DprE1 Inhibitors: Enduring Aspirations for Future Antituberculosis Drug Discovery.
32. Hybridization of the Pharmacophoric Features of Discoipyrrole C and Combretastatin A‐4 toward New Anticancer Leads.
33. Well‐Defined Anisotropic Self‐Assembly from Peptoids and Their Biomedical Applications.
34. Carborane‐Based Tebufelone Analogs and Their Biological Evaluation In Vitro.
35. Synthesis, Characterization and in vitro Anticancer Evaluation of 5‐Sulfinyl(sulfonyl)‐4‐arylsulfonyl‐Substituted 1,3‐Oxazoles.
36. Design, Synthesis, and Biological Evaluation of Histone Deacetylase Inhibitors Derived from Erianin and Its Derivatives.
37. Step‐Economical Mechanosynthesis of Hybrid Azoles: Deciphering Their π‐Orbital and Pharmacological Characteristics.
38. Evaluation of the Antiparasitic and Antifungal Activities of Synthetic Piperlongumine‐Type Cinnamide Derivatives: Booster Effect by Halogen Substituents.
39. Praziquantel – 50 Years of Research.
40. Structure‐Activity Relationships of Metal‐Based Inhibitors of the Mitochondrial Calcium Uniporter.
41. A Reinvestigation of the Role of the Sorbic Acid Tail on the Antibacterial and Anti‐Tuberculosis Properties of Moiramide B.
42. Not Every Hit‐Identification Technique Works on 1‐Deoxy‐d‐Xylulose 5‐Phosphate Synthase (DXPS): Making the Most of a Virtual Screening Campaign.
43. Versatile Diazomethane Sulfonamide for Expedited Exploration of Azole‐Based Carbonic Anhydrase Inhibitors via [3+2] Cycloaddition.
44. Development of Enterovirus Antiviral Agents That Target the Viral 2C Protein.
45. Scouting Different Phosphodiesterase 4 Inhibitor Chemotypes in Silico To Guide the Design of Anti‐inflammatory/Antioxidant Agents.
46. Design and Synthesis of 1,3‐Diynes as Potent Antifungal Agents against Aspergillus fumigatus.
47. Discovery of SI 1/20 and SI 1/22 as Mutual Prodrugs of 5‐Fluorouracil and Imidazole‐Based Heme Oxygenase 1 Inhibitor with Improved Cytotoxicity in DU145 Prostate Cancer Cells.
48. Recent Development of Copper (II) Complexes of Polypyridyl Ligands in Chemotherapy and Photodynamic Therapy.
49. Systematic Potency and Property Assessment of VHL Ligands and Implications on PROTAC Design.
50. Thiazolidinone‐Heterocycle Frameworks: A Concise Review of Their Pharmacological Significance.
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