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Review: [overview of the asymmetric synthesis of dihydrobenzoxazinone- and dihydroquinazolinone-based anti-HIV agents. [ABSTRACT FROM AUTHOR]

The reaction is environmentally benign. [ABSTRACT FROM AUTHOR]

The dual solvent-catalyst [bmim]OAc can be reused at least five times without an observable decrease in catalytic activity. [ABSTRACT FROM AUTHOR]

An abstract of the article "Efficient Synthesis of Quinazoline-2,4(1H,3H)-diones from CO2 and 2-Aminobenzonitriles in Water Without Any Catalyst" by J. Ma and colleagues is presented.

An efficient method for the asymmetric hydrogenation of fluorinated quinazolines (I) to chiral fluorinated dihydroquinazolines is developed using a Pd-SynPhos complex as catalyst. [ABSTRACT FROM AUTHOR]

An enantioselective aza-Friedel-Crafts reaction of cyclic N-acylketimines with electron-rich arenes is developed. [ABSTRACT FROM AUTHOR]

DPC 083 (X) is prepared in 5 steps starting from the enantiomer of Va. [ABSTRACT FROM AUTHOR]

The article presents chemical equations related to the article "Bisphosphine-Triggered One-Pot Sequential [3 + 2]/[3 + 2] Annulation of Allenoates with Cyclic Ketimines" by S. Wang, and others, published in the "Organic Letters" in 2013.

A series of N-fused tricyclic products are obtained under mild conditions. [ABSTRACT FROM AUTHOR]

This is the first hydrogen-bond-directed enantioselective decarboxylative Mannich reaction of β-ketoacids with ketimines affording quinazolinone derivatives with quaternary stereocenters in high yields and with excellent enantioselectivities using saccharide-based amino-thiourea organocatalysts. [ABSTRACT FROM AUTHOR]

The enantioselective Strecker reaction of ketimines (I) with trimethylsilyl cyanide is used for the preparation of quinazolinones (III). [ABSTRACT FROM AUTHOR]

The reaction proceeds well using a chiral chloramphenicol-amine derivative as catalyst. [ABSTRACT FROM AUTHOR]